SCHEMBL3288306

SCHEMBL3288306

Cc1cc(Nc2nc(-c3cc(CNC=O)ccc3F)cc3nccn23)n[nH]1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PLK4 O00444 9/20 0.40
NTRK1 P04629 9/20 0.40
MAP4K2 Q12851 1/20 0.39
PAK4 O96013 2/20 0.34
RET P07949 3/20 0.34
PI4KB Q9UBF8 1/20 0.33
AURKA O14965 1/20 0.33
AURKB Q96GD4 1/20 0.33
NTRK3 Q16288 1/20 0.32
NTRK2 Q16620 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3284835 0.87 PLK4 (0.40) PLK4NTRK1PAK4RETAURKA
SCHEMBL3288291 0.85 MAP4K2 (0.41) PLK4MAP4K2PAK4RETAURKA
SCHEMBL3033835 0.84 RET (0.47) PLK4NTRK1MAP4K2RETAURKA
SCHEMBL13221083 0.74 GSK3B (0.53) PLK4MAP4K2RETAURKAAURKB
SCHEMBL3028149 0.74 MAP4K2 (0.41) PLK4MAP4K2PAK4RETAURKA
SCHEMBL3285891 0.72 PAK1 (0.43) NTRK1
SCHEMBL13221158 0.72 NTRK1 (0.52) PLK4NTRK1PAK4AURKANTRK3
SCHEMBL5088382 0.72 MAP4K2 (0.64) PLK4MAP4K2RETAURKAAURKB
SCHEMBL13220904 0.72 ALK (0.49) PLK4MAP4K2RETAURKAAURKB
SCHEMBL3045180 0.72 RET (0.49) PLK4NTRK1RETAURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7713973-B2 Kinase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-05-11 US disclosed