SCHEMBL3285891

SCHEMBL3285891

O=CNCc1cccc(-c2cc3nccn3c(Nc3cc(C4CC4)[nH]n3)n2)c1

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PAK1 Q13153 1/20 0.43
IGF1R P08069 10/20 0.40
NTRK1 P04629 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13221081 0.87 PAK1 (0.44) PAK1IGF1RNTRK1
SCHEMBL3036860 0.87 PAK1 (0.42) PAK1IGF1RNTRK1
SCHEMBL3046927 0.87 SRC (0.42) PAK1IGF1RNTRK1
SCHEMBL3288291 0.86 MAP4K2 (0.41) IGF1R
SCHEMBL3045432 0.86 IGF1R (0.43) PAK1IGF1R
SCHEMBL3038521 0.85 WDR5 (0.45) PAK1IGF1R
SCHEMBL13220997 0.84 NEK1 (0.49) PAK1IGF1R
SCHEMBL3041108 0.84 PAK1 (0.40) PAK1IGF1R
SCHEMBL13221055 0.83 NEK1 (0.45) PAK1IGF1R
SCHEMBL3035000 0.83 PAK1 (0.40) PAK1IGF1RNTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7713973-B2 Kinase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-05-11 US disclosed