SCHEMBL3300767

SCHEMBL3300767

C=C[C@@H](Oc1ccc(C(F)(F)F)cc1)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 5/20 0.57
SLC6A4 P31645 6/20 0.54
SLC6A2 P23975 5/20 0.54
SLC6A3 Q01959 4/20 0.54
KCNK2 O95069 2/20 0.54
KCNH2 Q12809 2/20 0.54
CACNA1C Q13936 2/20 0.54
MEN1 O00255 4/20 0.50
KMT2A Q03164 4/20 0.50
LMNA P02545 4/20 0.50
HRH3 Q9Y5N1 2/20 0.50
NPC1 O15118 2/20 0.50
CYP2D6 P10635 2/20 0.50
CYP2C19 P33261 2/20 0.50
MTOR P42345 2/20 0.50
RAB9A P51151 2/20 0.50
CYP3A4 P08684 2/20 0.50
HTR2C P28335 2/20 0.50
TSHR P16473 2/20 0.50
KDM4E B2RXH2 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4865335 0.86 SRD5A2 (0.42) SLC7A5SLC6A4SLC6A2SLC6A3KCNK2
SCHEMBL8466535 0.83 SLC7A5 (0.40) SLC7A5SLC6A4SLC6A2SLC6A3KCNK2
SCHEMBL3291158 0.82 SLC6A4 (0.39) SLC7A5SLC6A4CYP2C19CYP3A4TSHR
SCHEMBL8163510 0.80 CYP1A2 (0.42) SLC7A5CYP2C19CYP3A4CYP1A2CYP2C9
SCHEMBL3299568 0.77 SLC6A4 (0.46) SLC7A5SLC6A4SLC6A2SLC6A3MEN1
SCHEMBL3294416 0.77 CA4 (0.46) MEN1KMT2ALMNANPC1RAB9A
SCHEMBL3295214 0.77 SLC6A4 (0.46) SLC6A4SLC6A2SLC6A3PPARGPPARA
SCHEMBL3294031 0.77 NPSR1 (0.41) SLC7A5MEN1KMT2ALMNATSHR
SCHEMBL7239564 0.77 SLC7A5 (0.68) SLC7A5SLC6A4SLC6A2SLC6A3KCNK2
SCHEMBL8625767 0.75 ALDH1A3 (0.50) KMT2ALMNARAB9AKDM4EDRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7732365-B2 Enantioselective amination and etherification YALE UNIVERSITY (US) 2010-06-08 US disclosed
US-20060199728-A1 Enantioselective amination and etherification YALE UNIVERSITY (US) 2006-09-07 US disclosed