SCHEMBL3324259

SCHEMBL3324259

CC(C)(C)OC(=O)N1CCC[C@H](COc2ccc(F)cc2Oc2ccccc2)C1

nearest known ligand 0.69

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.54
RBP4 P02753 3/20 0.49
HTR6 P50406 6/20 0.46
BCHE P06276 4/20 0.46
KAT7 O95251 1/20 0.46
KAT8 Q9H7Z6 1/20 0.46
ALOX5AP P20292 1/20 0.46
FEN1 P39748 1/20 0.46
ACKR3 P25106 1/20 0.46
CHEK2 O96017 1/20 0.46
CSF1R P07333 1/20 0.46
HCRTR1 O43613 1/20 0.44
HCRTR2 O43614 1/20 0.44
KDM1A O60341 1/20 0.44
BRD3 Q15059 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3324264 1.00 SCN9A (0.54) SCN9ARBP4HTR6BCHEKAT7
SCHEMBL3325117 0.85 SCN9A (0.58) SCN9ARBP4HTR6BCHEKAT7
SCHEMBL3325111 0.85 SCN9A (0.58) SCN9ARBP4HTR6BCHEKAT7
SCHEMBL8433798 0.85 SCN9A (0.52) SCN9ARBP4HTR6BCHEKAT7
SCHEMBL9901066 0.84 SCN9A (0.54) SCN9AKAT7KAT8ALOX5APFEN1
SCHEMBL27157955 0.84 SCN9A (0.55) SCN9ARBP4HTR6BCHEALOX5AP
SCHEMBL3443787 0.84 CHEK2 (0.56) SCN9AHTR6BCHEKAT7KAT8
SCHEMBL3443784 0.84 CHEK2 (0.56) SCN9AHTR6BCHEKAT7KAT8
SCHEMBL3321403 0.83 SCN9A (0.48) SCN9ARBP4HTR6BCHEALOX5AP
SCHEMBL3321410 0.83 SCN9A (0.48) SCN9ARBP4HTR6BCHEALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100120858-A1 Piperidine Derivatives PFIZER INC. 2010-05-13 US disclosed
EP-2066630-A1 PIPERIDINE DERIVATIVES Pfizer Products Incorporated (US) 2009-06-10 EP disclosed
WO-2008023258-A1 PIPERIDINE DERIVATIVES PFIZER PRODUCTS INC. (US) 2008-02-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100120858-A1 Piperidine Derivatives P2RX5, P2RX7, P2RX1 SCN9A 818/4885RBP4 2312/4885HTR6 832/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.