1,2,3,4-Tetrahydroisoquinoline

1,2,3,4-Tetrahydroisoquinoline

SCHEMBL3328852

c1ccc2[nH]ccc2c1.c1ccc2c(c1)CCNC2

nearest known ligand 0.66

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PNMT P11086 5/20 0.66
CD44 P16070 1/20 0.66
MAOB P27338 1/20 0.66
TRPA1 O75762 1/20 0.59
CA1 P00915 1/20 0.59
CA2 P00918 1/20 0.59
ITGB2 P05107 1/20 0.59
ICAM1 P05362 1/20 0.59
ITGAL P20701 1/20 0.59
CA4 P22748 1/20 0.59
CA6 P23280 1/20 0.59
AHR P35869 1/20 0.59
ADK P55263 1/20 0.59
HTR2C P28335 1/20 0.50
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
ASIC3 Q9UHC3 1/20 0.40
PRCP P42785 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
1,2,3,4-Tetrahydroisoquinoline SCHEMBL7327227 0.83 PNMT (0.86) PNMTCD44MAOBHTR2CADRA2A
1,2,3,4-Tetrahydroisoquinoline SCHEMBL29360217 0.81 PNMT (1.00) PNMTCD44MAOBHTR2CADRA2A
1,2,3,4-Tetrahydroisoquinoline SCHEMBL28236302 0.81 PNMT (1.00) PNMTCD44MAOBHTR2CADRA2A
1,2,3,4-Tetrahydroisoquinoline SCHEMBL19085 0.81 PNMT (1.00) PNMTCD44MAOBHTR2CADRA2A
1,2,3,4-Tetrahydroisoquinoline SCHEMBL4243903 0.79 PNMT (0.95) PNMTCD44MAOBHTR2CADRA2A
1,2,3,4-Tetrahydroisoquinoline SCHEMBL5411332 0.79 PNMT (0.95) PNMTCD44MAOBHTR2CADRA2A
1,2,3,4-Tetrahydroisoquinoline SCHEMBL2082936 0.79 PNMT (0.95) PNMTCD44MAOBHTR2CADRA2A
1,2,3,4-Tetrahydroisoquinoline SCHEMBL20524019 0.79 PNMT (0.95) PNMTCD44MAOBHTR2CADRA2A
SCHEMBL11838922 0.79 PNMT (0.95) PNMTCD44MAOBHTR2CADRA2A
1,2,3,4-Tetrahydroisoquinoline SCHEMBL11457582 0.79 PNMT (0.95) PNMTCD44MAOBHTR2CADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8362066-B2 Compounds and methods for treating protein folding disorders TREVENTIS CORPORATION (US) 2013-01-29 US disclosed
US-20100144821-A1 COMPOUNDS AND METHODS FOR TREATING PROTEIN FOLDING DISORDERS QUEEN'S UNIVERSITY AT KINGSTON (CA) 2010-06-10 US disclosed
EP-2081892-A1 COMPOUNDS AND METHODS FOR TREATING PROTEIN FOLDING DISORDERS Queen's University at Kingston (CA) 2009-07-29 EP disclosed
WO-2008058402-A1 COMPOUNDS AND METHODS FOR TREATING PROTEIN FOLDING DISORDERS QUEEN'S UNIVERSITY AT KINGSTON (CA) 2008-05-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100144821-A1 COMPOUNDS AND METHODS FOR TREATING PROTEIN FOLDING DISORDERS SNCA, MAPT, APP PNMT 627/4885CD44 2761/4885MAOB 841/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.