SCHEMBL333182

SCHEMBL333182

CNCCCN1CCc2cc(OC)c(OC)cc2CC1=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCN4 Q9Y3Q4 2/20 0.58
MAPT P10636 1/20 0.58
GAA P10253 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
SLC6A4 P31645 2/20 0.57
CYP3A4 P08684 1/20 0.57
ALOX15 P16050 1/20 0.57
CHRM2 P08172 1/20 0.57
HTR1A P08908 1/20 0.57
DRD3 P35462 1/20 0.57
KCNH2 Q12809 1/20 0.57
POLB P06746 1/20 0.45
PGK1 P00558 1/20 0.44
DRD1 P21728 1/20 0.44
DRD4 P21917 1/20 0.44
DRD5 P21918 1/20 0.44
MAOA P21397 2/20 0.42
MAOB P27338 2/20 0.42
ABCB1 P08183 2/20 0.42
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10597759 0.99 CYP3A4 (0.59) HCN4MAPTGAASMN1; SMN2SLC6A4
SCHEMBL14696925 0.89 GAA (0.68) HCN4MAPTGAASMN1; SMN2SLC6A4
SCHEMBL10978574 0.88 HCN4 (0.56) HCN4MAPTGAASMN1; SMN2SLC6A4
SCHEMBL15980993 0.85 GAA (0.62) HCN4MAPTGAASMN1; SMN2SLC6A4
SCHEMBL9624879 0.85 MEN1 (0.58) HCN4MAPTHTR1ADRD3DRD1
SCHEMBL9032662 0.84 GAA (0.61) HCN4MAPTGAASMN1; SMN2SLC6A4
SCHEMBL14696959 0.84 GAA (0.61) HCN4MAPTGAASMN1; SMN2SLC6A4
SCHEMBL30081993 0.84 GAA (0.61) HCN4MAPTGAASMN1; SMN2SLC6A4
SCHEMBL11094479 0.83 HCN4 (0.55) HCN4MAPTGAASMN1; SMN2SLC6A4
SCHEMBL9032571 0.83 HCN4 (0.60) HCN4MAPTGAASMN1; SMN2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113030328-B Method for detecting genotoxic impurities in ivabradine hydrochloride 北京阳光诺和药物研究股份有限公司 2023-03-14 CN disclosed
CN-113030328-A Method for detecting genotoxic impurities in ivabradine hydrochloride 北京阳光诺和药物研究股份有限公司 2021-06-25 CN disclosed
EP-2566850-B1 INDUSTRIAL PROCESS FOR THE SYNTHESIS OF IVABRADINE HYDROBROMIDE SALT RICHTER GEDEON NYRT (HU) 2018-04-11 EP disclosed
EP-2726462-B1 ACETONE SOLVATE OF IVABRADINE HYDROCHLORIDE SANDOZ AG (CH) 2017-03-22 EP disclosed
US-8415468-B2 Process for the synthesis of ivabradine and addition salts thereof with a pharmaceutically acceptable acid LES LABORATOIRES SERVIER (FR) 2013-04-09 US disclosed
EP-2202225-B1 New method for synthesising ivabradine and its added salts with a pharmaceutically acceptable acid. SERVIER LAB (FR) 2012-10-24 EP disclosed
US-8119794-B2 Process for the synthesis of ivabradine and addition salts thereof with a pharmaceutically acceptable acid LES LABORATOIRES SERVIER (FR) 2012-02-21 US disclosed
US-8119794-B2 Process for the synthesis of ivabradine and addition salts thereof with a pharmaceutically acceptable acid LES LABORATOIRES SERVIER (FR) 2012-02-21 US disclosed
US-8097720-B2 Process for the synthesis of ivabradine and addition salts thereof with a pharmaceutically acceptable acid Les Laboratories Server (FR) 2012-01-17 US disclosed
EP-2398802-A1 DERIVATIVES OF 6-CYCLOAMINO-2-THIENYL-3-(PYRIDIN-4-YL)IMIDAZO[1,2-b]-PYRIDAZINE AND 6-CYCLOAMINO-2-FURANYL-3-(PYRIDIN-4-YL)IMIDAZO[1,2-b]-PYRIDAZINE, PREPARATION AND THERAPEUTIC APPLICATION THEREOF SANOFI (FR) 2011-12-28 EP disclosed
EP-0109636-B1 BENZAZEPINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICAL COMPOUNDS Dr. Karl Thomae GmbH (DE) 1989-01-18 EP disclosed
US-4737495-A ANTIALLERGENS, ANTISCHEMIC, HYPOTENSIVE AGENTS DR. KARL TOMAE, GMBH (DE) 1988-04-12 US disclosed
EP-0259793-A1 Naphthyl derivatives, medicaments containing them and processes for their preparation Dr. Karl Thomae GmbH (DE) 1988-03-16 EP disclosed
EP-0204349-A2 Heteroaromatic amine derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1986-12-10 EP disclosed
US-4604389-A Benzazepine derivatives DR. KARL THOMAE GMBH (DE) 1986-08-05 US disclosed
EP-0161599-A2 Benzazepine derivatives, medicines containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1985-11-21 EP disclosed
EP-0065229-B1 BENZAZEPINES, PROCESS FOR THEIR PREPARATION AND THEIR APPLICATION AS PHARMACEUTICAL PREPARATIONS Dr. Karl Thomae GmbH (DE) 1985-08-07 EP disclosed
US-4490369-A HYPOTENSIVE, BRRADYCARDIAL DR. KARL THOMAE GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1984-12-25 US disclosed
EP-0109636-A2 Benzazepine derivatives, process for their preparation and their use as pharmaceutical compounds Dr. Karl Thomae GmbH (DE) 1984-05-30 EP disclosed
EP-0065229-A1 Benzazepines, process for their preparation and their application as pharmaceutical preparations Dr. Karl Thomae GmbH (DE) 1982-11-24 EP disclosed