SCHEMBL3345453

SCHEMBL3345453

COc1cc(N2CCC(O)CC2)ccc1N.COc1cc(N2CCC(O)CC2)ccc1N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTSR1 P30989 1/20 0.43
ALDH1A1 P00352 4/20 0.43
CYP3A4 P08684 2/20 0.43
TSHR P16473 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
LGMN Q99538 1/20 0.43
CHEK1 O14757 1/20 0.43
SUV39H2 Q9H5I1 1/20 0.43
DPP4 P27487 4/20 0.42
CDK1 P06493 1/20 0.42
CDK2 P24941 1/20 0.42
KDM4E B2RXH2 1/20 0.41
PDE7A Q13946 2/20 0.41
MAPT P10636 1/20 0.41
LMNA P02545 1/20 0.40
INSR P06213 1/20 0.40
IGF1R P08069 1/20 0.40
ALK Q9UM73 1/20 0.40
DCLK1 O15075 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL310068 1.00 NTSR1 (0.43) NTSR1ALDH1A1CYP3A4TSHRHSD17B10
SCHEMBL30682434 1.00 NTSR1 (0.43) NTSR1ALDH1A1CYP3A4TSHRHSD17B10
SCHEMBL10205069 0.92 ALK (0.43) NTSR1ALDH1A1LGMNCHEK1SUV39H2
SCHEMBL5406594 0.91 DPP4 (0.46) NTSR1ALDH1A1CYP3A4TSHRHSD17B10
Hydrochloric Acid SCHEMBL5387731 0.90 DPP4 (0.45) NTSR1ALDH1A1CYP3A4SUV39H2DPP4
SCHEMBL24073829 0.88 CHEK1 (0.46) NTSR1ALDH1A1CYP3A4LGMNCHEK1
SCHEMBL17265199 0.88 ALDH1A1 (0.46) ALDH1A1CYP3A4TSHRHSD17B10TDP1
SCHEMBL520117 0.87 SLC6A4 (0.40) NTSR1LGMNSUV39H2DPP4PDE7A
SCHEMBL519205 0.87 SLC6A4 (0.40) NTSR1LGMNSUV39H2DPP4PDE7A
SCHEMBL519204 0.87 SLC6A4 (0.40) NTSR1LGMNSUV39H2DPP4PDE7A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010049731-A1 PYRAZOLO- AND IMIDAZOPYRIDINYLPYRIMIDINEAMINES AS IGF-1R TYROSINE KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-05-06 WO disclosed