SCHEMBL3345829

SCHEMBL3345829

O=C(O)c1ccc(CCN2CCOCC2)n(Br)c1=O

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
MAPT P10636 3/20 0.42
KMT2A Q03164 3/20 0.42
POLB P06746 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
LMNA P02545 3/20 0.41
KDM4E B2RXH2 4/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
KDM4A O75164 1/20 0.40
MPI P34949 1/20 0.39
CYP2C19 P33261 1/20 0.39
TSHR P16473 1/20 0.39
GLA P06280 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6043506 0.71 ALDH1A1 (0.55) ALDH1A1MAPTKMT2APOLBSIGMAR1
SCHEMBL10426714 0.70 KMT2A (0.43) ALDH1A1MAPTKMT2APOLBSIGMAR1
SCHEMBL10426713 0.69 KMT2A (0.43) ALDH1A1MAPTKMT2APOLBSIGMAR1
SCHEMBL16411512 0.69 ALDH1A1 (0.44) ALDH1A1MAPTKMT2APOLBSIGMAR1
SCHEMBL12805538 0.68 CNR1 (0.43) ALDH1A1MAPTKMT2AKDM4EKDM4A
SCHEMBL10425888 0.68 POLB (0.48) ALDH1A1MAPTKMT2APOLBSIGMAR1
SCHEMBL4929767 0.68 KLK7 (0.42) ALDH1A1MAPTKMT2APOLBSIGMAR1
SCHEMBL10426684 0.68 POLB (0.47) ALDH1A1MAPTKMT2APOLBSIGMAR1
SCHEMBL10425887 0.68 POLB (0.47) ALDH1A1MAPTKMT2APOLBSIGMAR1
SCHEMBL3373579 0.67 PARP1 (0.50) ALDH1A1MAPTKMT2APOLBSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038081-A2 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB (SE) 2010-04-08 WO disclosed