SCHEMBL3346070

SCHEMBL3346070

Cc1cc2c(ccc3nnnn32)c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.43
PTGS1 P23219 4/20 0.39
PTGS2 P35354 3/20 0.39
ABCB1 P08183 5/20 0.39
AKR1C3 P42330 2/20 0.39
AKR1C2 P52895 2/20 0.39
PTGDR2 Q9Y5Y4 6/20 0.37
MEN1 O00255 2/20 0.37
LMNA P02545 2/20 0.37
CYP1A2 P05177 2/20 0.37
MAPT P10636 2/20 0.37
CYP2C9 P11712 2/20 0.37
PMP22 Q01453 2/20 0.37
KMT2A Q03164 2/20 0.37
HIF1A Q16665 2/20 0.37
PTGES O14684 1/20 0.37
ABCC3 O15438 1/20 0.37
ABCC4 O15439 1/20 0.37
ABCB11 O95342 1/20 0.37
MT-CO2 P00403 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20021162 0.82 KDM4E (0.43) KDM4EPTGS1PTGS2ABCB1AKR1C3
SCHEMBL10284225 0.78 KDM4E (0.44) KDM4EPTGS1PTGS2ABCB1AKR1C3
SCHEMBL252572 0.75 CYP3A4 (0.45) CYP3A4
SCHEMBL20021131 0.74 PTGDR2 (0.47) KDM4EPTGS1PTGS2ABCB1PTGDR2
SCHEMBL15182648 0.73 CYP3A4 (0.38) CYP3A4
SCHEMBL3297610 0.73 KDM4E (0.54) KDM4EPTGDR2MEN1LMNAKMT2A
SCHEMBL252269 0.72 HPGD (0.32) ALDH1A1CYP3A4TSHR
SCHEMBL252268 0.72 HPGD (0.32) ALDH1A1CYP3A4TSHR
SCHEMBL3303954 0.72 KDM4E (0.53) KDM4EPTGDR2MEN1LMNAMAPT
SCHEMBL18892276 0.72 KDM4E (0.47) KDM4EPTGDR2MEN1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012003498-A1 2 -QUINOLINYL- ACETIC ACID DERIVATIVES AS HIV ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2012-01-05 WO disclosed