SCHEMBL3346263

SCHEMBL3346263

C#Cc1ccc(CCN[C@H](CC(C)C)C(=O)OC2CCCC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 7/20 0.48
MAPK13 O15264 1/20 0.48
MAPK12 P53778 1/20 0.48
MAPK11 Q15759 1/20 0.48
NPR3 P17342 1/20 0.41
ACACB O00763 3/20 0.39
MMP2 P08253 2/20 0.38
MMP9 P14780 2/20 0.38
ANPEP P15144 2/20 0.38
LTA4H P09960 1/20 0.38
LAP3 P28838 1/20 0.38
NPEPPS P55786 1/20 0.38
ERAP2 Q6P179 1/20 0.38
ERAP1 Q9NZ08 1/20 0.38
TPSAB1 Q15661 1/20 0.36
TPSD1 Q9BZJ3 1/20 0.36
TPSG1 Q9NRR2 1/20 0.36
CYP19A1 P11511 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3346257 1.00 MAPK14 (0.48) MAPK14MAPK13MAPK12MAPK11NPR3
SCHEMBL561106 0.89 NPR3 (0.42) MAPK14MAPK13MAPK12MAPK11NPR3
SCHEMBL561107 0.89 NPR3 (0.42) MAPK14MAPK13MAPK12MAPK11NPR3
SCHEMBL2280856 0.86 MAPK14 (0.50) MAPK14MAPK13MAPK12MAPK11NPR3
SCHEMBL2280854 0.86 MAPK14 (0.50) MAPK14MAPK13MAPK12MAPK11NPR3
SCHEMBL3345198 0.85 MAPK14 (0.48) MAPK14MAPK13MAPK12MAPK11NPR3
SCHEMBL3345202 0.85 MAPK14 (0.48) MAPK14MAPK13MAPK12MAPK11NPR3
SCHEMBL2276180 0.81 MAPK14 (0.45) MAPK14MAPK13MAPK12MAPK11NPR3
SCHEMBL2276175 0.81 MAPK14 (0.45) MAPK14MAPK13MAPK12MAPK11NPR3
SCHEMBL3344769 0.78 ACACB (0.41) ACACBTPSAB1TPSD1TPSG1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010043865-A1 INHIBITORS OF HSP90 CHROMA THERAPEUTICS LTD (GB) 2010-04-22 WO disclosed