SCHEMBL3344769

SCHEMBL3344769

C#Cc1ccc(CN[C@@H](C)C(=O)OC2CCCC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACACB O00763 11/20 0.41
PDK1 Q15118 1/20 0.41
CYP19A1 P11511 1/20 0.40
TPSAB1 Q15661 2/20 0.39
TPSD1 Q9BZJ3 2/20 0.39
TPSG1 Q9NRR2 2/20 0.39
ALDH1A1 P00352 1/20 0.39
ALOX12 P18054 1/20 0.39
HRH1 P35367 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
GRIN2B Q13224 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL561107 0.86 NPR3 (0.42) ACACBCYP19A1TPSAB1TPSD1TPSG1
SCHEMBL561106 0.86 NPR3 (0.42) ACACBCYP19A1TPSAB1TPSD1TPSG1
SCHEMBL13424284 0.86 MEP1B (0.38) PDK1CYP19A1ALDH1A1
SCHEMBL3345164 0.84 ACACB (0.43) ACACBPDK1CYP19A1TPSAB1TPSD1
SCHEMBL3346269 0.84 PDK1 (0.42) PDK1CYP19A1TPSAB1TPSD1TPSG1
SCHEMBL8313235 0.82 F2 (0.49) CYP19A1
SCHEMBL8313233 0.82 F2 (0.49) CYP19A1
SCHEMBL1491397 0.78 CACNA1B (0.49) PDK1TPSAB1TPSD1TPSG1ALDH1A1
SCHEMBL1491399 0.78 CACNA1B (0.49) PDK1TPSAB1TPSD1TPSG1ALDH1A1
SCHEMBL3346257 0.78 MAPK14 (0.48) ACACBCYP19A1TPSAB1TPSD1TPSG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010043865-A1 INHIBITORS OF HSP90 CHROMA THERAPEUTICS LTD (GB) 2010-04-22 WO disclosed
WO-2010043865-A1 INHIBITORS OF HSP90 CHROMA THERAPEUTICS LTD (GB) 2010-04-22 WO disclosed