SCHEMBL3346355

SCHEMBL3346355

Cc1csc(-c2cc(N)cs2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.47
NOS1 P29475 2/20 0.47
PLAU P00749 1/20 0.41
PDE10A Q9Y233 1/20 0.40
CYP3A4 P08684 2/20 0.39
CYP2E1 P05181 1/20 0.39
CYP2A6 P11509 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2B6 P20813 1/20 0.39
SRC P12931 1/20 0.37
CDK2 P24941 1/20 0.37
ZAP70 P43403 1/20 0.37
SYK P43405 1/20 0.37
RAB9A P51151 4/20 0.37
GAA P10253 3/20 0.37
KMT2A Q03164 3/20 0.37
NPC1 O15118 3/20 0.37
MAPK1 P28482 2/20 0.37
GLA P06280 1/20 0.36
MEN1 O00255 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18157874 0.73 SMN1; SMN2 (0.55) SMN1; SMN2NOS1PLAUPDE10ACYP3A4
SCHEMBL13680611 0.71 CYP3A4 (0.51) SMN1; SMN2NOS1PDE10ACYP3A4CYP2E1
SCHEMBL1822397 0.70 SMN1; SMN2 (0.44) SMN1; SMN2NOS1PLAUPDE10ACYP3A4
SCHEMBL13680759 0.70 BACE1 (0.49) SMN1; SMN2NOS1PLAUPDE10ACYP3A4
SCHEMBL19853525 0.69 ATP4A (0.38) SMN1; SMN2NOS1PLAUPDE10ACYP3A4
SCHEMBL18175150 0.69 TSHR (0.57) SMN1; SMN2NOS1PDE10ACYP3A4CYP2E1
SCHEMBL17407204 0.68 SMN1; SMN2 (0.68) SMN1; SMN2NOS1PDE10ACYP3A4CYP2E1
SCHEMBL890218 0.68 NPC1 (0.50) SMN1; SMN2NOS1PLAUPDE10ACYP3A4
SCHEMBL28996037 0.68 PDE10A (0.42) SMN1; SMN2NOS1PLAUPDE10ACYP3A4
SCHEMBL996759 0.68 SMN1; SMN2 (0.45) SMN1; SMN2NOS1PLAUPDE10ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010045008-A1 AMIDES OF THIENO[2,3-d]PYRIMIDINE AND THEIR USE AS ADENOSINE A2a RECEPTOR ANTAGONISTS JANSSEN PHARMACEUTICA NV (BE) 2010-04-22 WO disclosed