SCHEMBL3346572

SCHEMBL3346572

C[C@H](NC(=O)[C@@H]1CNC[C@H]1c1ccc(C(F)(F)F)cn1)c1cccc(F)c1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.51
PDE2A O00408 2/20 0.39
MAPK1 P28482 2/20 0.38
ROCK2 O75116 6/20 0.38
ACACB O00763 1/20 0.37
KIT P10721 3/20 0.37
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
JAK3 P52333 1/20 0.37
CASR P41180 1/20 0.37
ROCK1 Q13464 3/20 0.36
OPRM1 P35372 1/20 0.36
OPRL1 P41146 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3346217 0.91 KCNH2 (0.51) KCNH2PDE2AACACBKIT
SCHEMBL3346383 0.90 KCNH2 (0.50) KCNH2PDE2AMAPK1ROCK2ACACB
SCHEMBL13365135 0.90 KCNH2 (0.57) KCNH2PDE2AACACB
SCHEMBL3346567 0.89 KCNH2 (0.59) KCNH2PDE2AMAPK1ACACB
SCHEMBL3350854 0.89 KCNH2 (0.49) KCNH2MAPK1ROCK2ROCK1
SCHEMBL3380842 0.87 KCNH2 (0.40) KCNH2MAPK1ROCK2KITJAK2
SCHEMBL13365111 0.86 KCNH2 (0.68) KCNH2PDE2AROCK2CASROPRM1
SCHEMBL3350659 0.86 KCNH2 (0.68) KCNH2PDE2AROCK2CASROPRM1
SCHEMBL3346554 0.83 KCNH2 (0.48) KCNH2PDE2AROCK2ACACBROCK1
SCHEMBL3347928 0.82 KCNH2 (0.53) KCNH2MAPK1ROCK2KITJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed