SCHEMBL3350854

SCHEMBL3350854

COc1cccc([C@H](C)NC(=O)[C@@H]2CNC[C@H]2c2ccc(C(F)(F)F)cn2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.49
POLB P06746 2/20 0.48
MEN1 O00255 1/20 0.48
LMNA P02545 1/20 0.48
HTT P42858 1/20 0.48
KMT2A Q03164 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
ROCK2 O75116 15/20 0.46
PRKG1 Q13976 9/20 0.46
ROCK1 Q13464 10/20 0.43
PRKACA P17612 5/20 0.41
CYP2C9 P11712 3/20 0.41
GSK3A P49840 3/20 0.41
GSK3B P49841 3/20 0.41
PRKX P51817 3/20 0.41
CYP3A4 P08684 3/20 0.41
PRKACG P22612 2/20 0.41
PRKACB P22694 2/20 0.41
AKT1 P31749 2/20 0.41
CYP2D6 P10635 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3346217 0.89 KCNH2 (0.51) KCNH2
SCHEMBL3346572 0.89 KCNH2 (0.51) KCNH2ROCK2ROCK1MAPK1
SCHEMBL3346383 0.88 KCNH2 (0.50) KCNH2ROCK2ROCK1MAPK1
SCHEMBL13365135 0.87 KCNH2 (0.57) KCNH2
SCHEMBL3346689 0.87 POLB (0.50) POLBMEN1LMNAHTTKMT2A
SCHEMBL3346490 0.87 KCNH2 (0.65) KCNH2POLBMEN1LMNAHTT
SCHEMBL3346552 0.83 KCNH2 (0.45) KCNH2ROCK2ROCK1
SCHEMBL3346506 0.83 KCNH2 (0.51) KCNH2POLBMEN1LMNAHTT
SCHEMBL3346567 0.83 KCNH2 (0.59) KCNH2KMT2AMAPK1
SCHEMBL3347178 0.80 KCNH2 (0.53) KCNH2POLBMEN1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed