SCHEMBL3346554

SCHEMBL3346554

C[C@H](NC(=O)[C@@H]1CNC[C@H]1c1ccc(C(F)(F)F)cn1)c1ccccc1F

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.48
SSTR4 P31391 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37
NCOR2 Q9Y618 1/20 0.37
PDE2A O00408 6/20 0.37
ROCK2 O75116 3/20 0.35
ROCK1 Q13464 3/20 0.35
HCRTR1 O43613 1/20 0.35
ACACB O00763 1/20 0.35
TRPM8 Q7Z2W7 1/20 0.34
MC4R P32245 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13365135 0.87 KCNH2 (0.57) KCNH2PDE2AACACB
SCHEMBL13365050 0.87 SSTR4 (0.39) KCNH2SSTR4ROCK2ROCK1MC4R
SCHEMBL13365134 0.85 KCNH2 (0.64) KCNH2SSTR4PDE2ATRPM8MC4R
SCHEMBL3346452 0.85 KCNH2 (0.48) KCNH2SSTR4PDE2AROCK2ACACB
SCHEMBL3346567 0.85 KCNH2 (0.59) KCNH2PDE2AACACB
SCHEMBL3346572 0.83 KCNH2 (0.51) KCNH2PDE2AROCK2ROCK1ACACB
SCHEMBL3353119 0.81 KCNH2 (0.47) KCNH2SSTR4PDE2AACACB
SCHEMBL3346217 0.81 KCNH2 (0.51) KCNH2SSTR4PDE2AACACB
SCHEMBL3345898 0.81 KCNH2 (0.54) KCNH2SSTR4HDAC4ROCK2ROCK1
SCHEMBL3346383 0.81 KCNH2 (0.50) KCNH2PDE2AROCK2ROCK1ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed