SCHEMBL3346602

SCHEMBL3346602

Fc1cc(F)cc(Nc2nc(Cl)nc(NC3CCCC3)n2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSV O60911 2/20 0.70
PLAT P00750 2/20 0.70
CTSL P07711 2/20 0.70
CTSH P09668 2/20 0.70
CTSS P25774 2/20 0.70
CASP14 P31944 2/20 0.70
CTSK P43235 2/20 0.70
CASP6 P55212 2/20 0.70
CTSZ Q9UBR2 2/20 0.70
CTSB P07858 1/20 0.70
CASP4 P49662 1/20 0.70
CASP5 P51878 1/20 0.70
RAB9A P51151 1/20 0.61
PDE4A P27815 1/20 0.54
IDH1 O75874 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5031260 0.85 RAB9A (0.62) CTSVPLATCTSLCTSHCTSS
SCHEMBL3347831 0.82 CTSS (1.00) CTSVPLATCTSLCTSHCTSS
SCHEMBL14600703 0.78 RAB9A (0.75) CTSVPLATCTSLCTSHCTSS
SCHEMBL20938665 0.78 RAB9A (0.75) CTSVPLATCTSLCTSHCTSS
SCHEMBL3503380 0.78 RAB9A (0.80) CTSVPLATCTSLCTSHCTSS
SCHEMBL13326008 0.78 RAB9A (0.75) CTSVPLATCTSLCTSHCTSS
SCHEMBL5029172 0.78 RAB9A (0.70) CTSVPLATCTSLCTSHCTSS
SCHEMBL14294391 0.78 RAB9A (0.62) CTSVPLATCTSLCTSHCTSS
SCHEMBL20402878 0.78 PDE4A (0.82) CTSSCTSKRAB9APDE4A
SCHEMBL18557113 0.78 PDE4A (0.82) CTSSCTSKRAB9APDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059418-A1 SUBSTITUTED TRIAZINE AND PURINE COMPOUNDS, METHODS OF INHIBITING CRUZAIN AND RHODESAIN AND METHODS OF TREATING CHAGAS DISEASE AND AFRICAN TRYPANOSOMIASIS THE GOVERNMENT OF THE U.S.A. AS REPRESENTED BY THE SECRETARY OF THE DEPT. OF HEALTH & HUMAN SERVICES (US) 2010-05-27 WO disclosed
WO-2010059418-A1 SUBSTITUTED TRIAZINE AND PURINE COMPOUNDS, METHODS OF INHIBITING CRUZAIN AND RHODESAIN AND METHODS OF TREATING CHAGAS DISEASE AND AFRICAN TRYPANOSOMIASIS THE GOVERNMENT OF THE U.S.A. AS REPRESENTED BY THE SECRETARY OF THE DEPT. OF HEALTH & HUMAN SERVICES (US) 2010-05-27 WO disclosed