SCHEMBL3346870

SCHEMBL3346870

COc1ccccc1[C@H](C)NC(=O)[C@@H]1CNC[C@H]1c1ccc(C(F)(F)F)cc1

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.62
PDE2A O00408 1/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
SSTR4 P31391 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
FFAR1 O14842 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
MC4R P32245 4/20 0.38
CHRNA7 P36544 1/20 0.38
CCR3 P51677 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13365134 0.88 KCNH2 (0.64) KCNH2PDE2ASSTR4CYP3A4CYP2D6
SCHEMBL3346321 0.84 KCNH2 (0.77) KCNH2PDE2AHPGDCYP3A4CYP2D6
SCHEMBL3353100 0.82 KCNH2 (0.68) KCNH2PDE2ASMN1; SMN2CYP3A4CYP2D6
SCHEMBL3346490 0.82 KCNH2 (0.65) KCNH2PDE2ASMN1; SMN2CYP3A4CYP2D6
SCHEMBL3346026 0.81 KCNH2 (0.58) KCNH2SSTR4CYP3A4CYP2D6CYP2C9
SCHEMBL13365111 0.78 KCNH2 (0.68) KCNH2PDE2ACYP3A4CYP2D6CYP2C9
SCHEMBL3346364 0.78 KCNH2 (0.68) KCNH2PDE2ACYP3A4CYP2D6CYP2C9
SCHEMBL3350659 0.78 KCNH2 (0.68) KCNH2PDE2ACYP3A4CYP2D6CYP2C9
SCHEMBL3346599 0.78 KCNH2 (0.68) KCNH2PDE2ACYP3A4CYP2D6CYP2C9
SCHEMBL13365108 0.78 KCNH2 (0.64) KCNH2CYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed