SCHEMBL3348200

SCHEMBL3348200

COc1cccc([C@H](C)NC(=O)[C@@H]2CNC[C@H]2c2ccc(OC(F)(F)F)cc2)c1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.52
POLB P06746 2/20 0.51
ROCK2 O75116 7/20 0.49
PRKG1 Q13976 3/20 0.49
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
LMNA P02545 1/20 0.44
HTT P42858 1/20 0.44
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
GPR139 Q6DWJ6 4/20 0.41
ROCK1 Q13464 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3346914 0.90 KCNH2 (0.52) KCNH2POLBROCK2PRKG1GPR139
SCHEMBL3346490 0.90 KCNH2 (0.65) KCNH2POLBROCK2PRKG1MEN1
SCHEMBL3353031 0.88 KCNH2 (0.59) KCNH2ROCK2GPR139
SCHEMBL3347178 0.87 KCNH2 (0.53) KCNH2POLBROCK2PRKG1MEN1
SCHEMBL3348185 0.87 POLB (0.53) KCNH2POLBROCK2PRKG1MEN1
SCHEMBL3346274 0.87 POLB (0.54) KCNH2POLBROCK2PRKG1MEN1
SCHEMBL3346506 0.84 KCNH2 (0.51) KCNH2POLBROCK2PRKG1MEN1
SCHEMBL3353232 0.83 POLB (0.53) KCNH2POLBROCK2PRKG1MEN1
SCHEMBL3347954 0.83 POLB (0.54) KCNH2POLBROCK2PRKG1MEN1
SCHEMBL3412005 0.82 KCNH2 (0.55) KCNH2KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed