SCHEMBL3347178

SCHEMBL3347178

COc1cccc([C@H](C)NC(=O)[C@@H]2CNC[C@H]2c2ccc(C(C)(C)C)cc2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.53
POLB P06746 2/20 0.53
ROCK2 O75116 13/20 0.50
PRKG1 Q13976 9/20 0.50
SMN1; SMN2 Q16637 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
LMNA P02545 2/20 0.43
HTT P42858 2/20 0.43
ROCK1 Q13464 4/20 0.42
MAPK1 P28482 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CHEK1 O14757 1/20 0.42
RPS6KA5 O75582 1/20 0.42
PRKCG P05129 1/20 0.42
CDK1 P06493 1/20 0.42
PRKACA P17612 1/20 0.42
RPS6KB1 P23443 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3346490 0.91 KCNH2 (0.65) KCNH2POLBROCK2PRKG1SMN1; SMN2
SCHEMBL3346274 0.88 POLB (0.54) KCNH2POLBROCK2PRKG1SMN1; SMN2
SCHEMBL3348200 0.87 KCNH2 (0.52) KCNH2POLBROCK2PRKG1SMN1; SMN2
SCHEMBL3348185 0.86 POLB (0.53) KCNH2POLBROCK2PRKG1SMN1; SMN2
SCHEMBL3346485 0.86 KCNH2 (0.63) KCNH2LMNA
SCHEMBL3353232 0.85 POLB (0.53) KCNH2POLBROCK2PRKG1SMN1; SMN2
SCHEMBL3347954 0.84 POLB (0.54) KCNH2POLBROCK2PRKG1SMN1; SMN2
SCHEMBL3353100 0.82 KCNH2 (0.68) KCNH2POLBROCK2PRKG1SMN1; SMN2
SCHEMBL3352431 0.82 ROCK2 (0.52) KCNH2POLBROCK2PRKG1SMN1; SMN2
SCHEMBL3346506 0.82 KCNH2 (0.51) KCNH2POLBROCK2PRKG1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed