SCHEMBL3346914

SCHEMBL3346914

C[C@H](NC(=O)[C@@H]1CNC[C@H]1c1ccc(OC(F)(F)F)cc1)c1cccc(F)c1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.52
OPRM1 P35372 1/20 0.43
ROCK2 O75116 3/20 0.41
PDE2A O00408 2/20 0.39
GPR139 Q6DWJ6 2/20 0.39
KCNQ3 O43525 2/20 0.39
KCNQ2 O43526 2/20 0.39
HTR2C P28335 1/20 0.38
KCNQ4 P56696 1/20 0.38
KCNQ5 Q9NR82 1/20 0.38
POLB P06746 1/20 0.38
MC4R P32245 1/20 0.38
MC5R P33032 1/20 0.38
MC3R P41968 1/20 0.38
PRKG1 Q13976 1/20 0.37
ACACB O00763 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3348200 0.90 KCNH2 (0.52) KCNH2ROCK2GPR139POLBPRKG1
SCHEMBL3353031 0.89 KCNH2 (0.59) KCNH2ROCK2PDE2AGPR139KCNQ3
SCHEMBL3350659 0.87 KCNH2 (0.68) KCNH2OPRM1ROCK2PDE2AKCNQ3
SCHEMBL13365111 0.87 KCNH2 (0.68) KCNH2OPRM1ROCK2PDE2AKCNQ3
SCHEMBL13365065 0.85 KCNH2 (0.52) KCNH2ROCK2KCNQ3KCNQ2KCNQ4
SCHEMBL3353036 0.85 KCNH2 (0.52) KCNH2ROCK2KCNQ3KCNQ2KCNQ4
SCHEMBL13365099 0.85 KCNH2 (0.52) KCNH2ROCK2KCNQ3KCNQ2KCNQ4
SCHEMBL3353124 0.85 KCNH2 (0.52) KCNH2ROCK2KCNQ3KCNQ2KCNQ4
SCHEMBL3353040 0.82 KCNH2 (0.48) KCNH2ROCK2KCNQ3KCNQ2KCNQ4
SCHEMBL3347928 0.81 KCNH2 (0.53) KCNH2ROCK2KCNQ3KCNQ2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed