SCHEMBL3351417

SCHEMBL3351417

COc1cccc(CN(C[C@@H](O)[C@@H](N)Cc2ccccc2)C(=O)O)c1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGES O14684 5/20 0.47
TAAR1 Q96RJ0 2/20 0.46
TAS2R14 Q9NYV8 2/20 0.46
TSHR P16473 2/20 0.46
LPAR1 Q92633 1/20 0.45
LPAR5 Q9H1C0 1/20 0.45
CALM1 P0DP23 1/20 0.44
CAMKK2 Q96RR4 1/20 0.44
TSPO P30536 1/20 0.44
ALOX5 P09917 1/20 0.44
CETP P11597 1/20 0.43
HSD17B2 P37059 1/20 0.43
SLC2A1 P11166 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4666757 0.99 PTGES (0.47) PTGESTAAR1TAS2R14TSHRLPAR1
SCHEMBL4799435 0.91 BACE1 (0.44) PTGESTAAR1LPAR1LPAR5
SCHEMBL3881006 0.88 LTA4H (0.44) PTGESTAAR1TSHRTSPOALOX5
SCHEMBL5206234 0.88 LTA4H (0.44) PTGESTAAR1TSHRTSPOALOX5
SCHEMBL3877346 0.87 PTGES (0.43) PTGESTAAR1TAS2R14TSPOALOX5
SCHEMBL3877090 0.87 PTGES (0.43) PTGESTAAR1TAS2R14TSPOALOX5
SCHEMBL3877094 0.87 PTGES (0.43) PTGESTAAR1TAS2R14TSPOALOX5
SCHEMBL8347358 0.85 KMT2A (0.52) TAAR1CALM1CAMKK2CETP
SCHEMBL8125895 0.85 KMT2A (0.52) TAAR1CALM1CAMKK2CETP
SCHEMBL5130716 0.85 SLC2A1 (0.45) PTGESTAAR1SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7727997-B2 N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives ELAN PHARMACEUTICALS, INC. (US) 2010-06-01 US disclosed
US-20070213316-A1 Compounds that are effective inhibitors of beta-secretase; inhibitors of beta-secretase-mediated cleavage of amyloid precursor proteins; effective inhibitors of A beta production, and/or are effective to reduce amyloid beta deposits or plaques; treatment of disorders such as Alzheimer's Disease ELAN PHARMACEUTICALS, INC. 2007-09-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070213316-A1 Compounds that are effective inhibitors of beta-secretase; inhibitors of beta-secretase-mediated cleavage of amyloid precursor proteins; effective inhibitors of A beta production, and/or are effective to reduce amyloid beta deposits or plaques; treatment of disorders such as Alzheimer's Disease BACE1, BACE2, APP PTGES 1409/4885TAAR1 3168/4885TAS2R14 4471/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.