Phthalimide

Phthalimide

SCHEMBL335240

CC=O.O=C1NC(=O)c2ccccc21

nearest known ligand 0.75

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.75
CASP3 P42574 2/20 0.62
CASP7 P55210 2/20 0.62
CASP6 P55212 2/20 0.62
CASP8 Q14790 2/20 0.62
CASP2 P42575 1/20 0.62
SMN1; SMN2 Q16637 5/20 0.50
LMNA P02545 5/20 0.50
MAPK1 P28482 2/20 0.50
HSD17B10 Q99714 1/20 0.50
PARP1 P09874 3/20 0.48
PDGFRA P16234 1/20 0.48
FER P16591 1/20 0.48
LTK P29376 1/20 0.48
CDK8 P49336 1/20 0.48
ACVR1 Q04771 1/20 0.48
LRRK2 Q5S007 1/20 0.48
DYRK1B Q9Y463 1/20 0.48
PARP2 Q9UGN5 1/20 0.47
TDP2 O95551 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phthalimide SCHEMBL28635005 0.90 GSK3B (0.75) GSK3BCASP3CASP7CASP6CASP8
Phthalimide SCHEMBL28967086 0.88 GSK3B (0.71) GSK3BCASP3CASP7CASP6CASP8
Phthalimide SCHEMBL23063638 0.87 GSK3B (0.88) GSK3BCASP3CASP7CASP6CASP8
Phthalimide SCHEMBL29366030 0.87 GSK3B (1.00) GSK3BCASP3CASP7CASP6CASP8
Phthalimide SCHEMBL10192661 0.87 GSK3B (1.00) GSK3BCASP3CASP7CASP6CASP8
Phthalimide SCHEMBL7771670 0.87 GSK3B (1.00) GSK3BCASP3CASP7CASP6CASP8
Phthalimide SCHEMBL30125197 0.87 GSK3B (1.00) GSK3BCASP3CASP7CASP6CASP8
Phthalimide SCHEMBL11040503 0.87 GSK3B (1.00) GSK3BCASP3CASP7CASP6CASP8
Phthalimide SCHEMBL64 0.87 GSK3B (1.00) GSK3BCASP3CASP7CASP6CASP8
Phthalimide SCHEMBL28626273 0.86 GSK3B (0.68) GSK3BCASP3CASP7CASP6CASP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113956166-A Method for producing aminoacetaldehyde dimethyl acetal 上海鸣谦化工技术服务中心 2022-01-21 CN claimed
CN-113956166-A Method for producing aminoacetaldehyde dimethyl acetal 上海鸣谦化工技术服务中心 2022-01-21 CN disclosed
CN-113956166-A Method for producing aminoacetaldehyde dimethyl acetal 上海鸣谦化工技术服务中心 2022-01-21 CN disclosed
US-8097708-B2 10a-Azalide compound TAISHO PHARMACEUTICAL CO., LTD. (JP) 2012-01-17 US disclosed
US-20090281292-A1 10a-Azalide Compound MEIJI SEIKA PHARMA CO., LTD. (JP) 2009-11-12 US disclosed
EP-1985620-A1 10a-AZALIDE COMPOUND TAISHO PHARMACEUTICAL CO., LTD (JP) 2008-10-29 EP disclosed
US-6300316-B1 ANTIBIOTICS AS BACTERICIDE PFIZER INC 2001-10-09 US disclosed
US-6025350-A C-4\" substituted macrolide antibiotics PFIZER INC. (US) 2000-02-15 US disclosed
EP-0895999-A1 C-4\" substituted macrolide antibiotics Pfizer Products Inc. (US) 1999-02-10 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090281292-A1 10a-Azalide Compound IL17A, AZI2, HDAC9 GSK3B 2455/4885CASP3 1314/4885CASP7 277/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.