SCHEMBL3353241

SCHEMBL3353241

C[C@@H](Cc1ccc(Cl)cc1)NC(=O)[C@@H]1CNC[C@H]1c1ccc(C(F)(F)F)cc1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 8/20 0.59
MC4R P32245 9/20 0.47
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
MC5R P33032 2/20 0.42
MC3R P41968 2/20 0.42
ACACB O00763 1/20 0.41
MC1R Q01726 1/20 0.41
CNR2 P34972 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3346440 1.00 KCNH2 (0.59) KCNH2MC4RCYP3A4CYP2D6CYP2C9
SCHEMBL3346210 0.90 KCNH2 (0.59) KCNH2MC4RCYP3A4CYP2D6CYP2C9
SCHEMBL3346354 0.77 KCNH2 (0.67) KCNH2MC4R
SCHEMBL3353009 0.77 KCNH2 (0.67) KCNH2MC4R
SCHEMBL3350686 0.77 KCNH2 (0.63) KCNH2MC4RCYP3A4CYP2D6CYP2C9
SCHEMBL13365064 0.76 ACACB (0.47) ACACB
SCHEMBL3346321 0.76 KCNH2 (0.77) KCNH2MC4RCYP3A4CYP2D6CYP2C9
SCHEMBL13365134 0.73 KCNH2 (0.64) KCNH2MC4RCYP3A4CYP2D6CYP2C9
SCHEMBL13365108 0.73 KCNH2 (0.64) KCNH2MC4RCYP3A4CYP2D6CYP2C9
SCHEMBL3353012 0.73 KCNH2 (0.59) KCNH2MC4RCYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed