SCHEMBL3346210

SCHEMBL3346210

C[C@H](Cc1ccccc1)NC(=O)[C@@H]1CNC[C@H]1c1ccc(C(F)(F)F)cc1

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 8/20 0.59
MC4R P32245 2/20 0.48
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
MAOA P21397 1/20 0.43
TACR1 P25103 3/20 0.43
FFAR1 O14842 1/20 0.41
FPR2 P25090 1/20 0.41
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3353241 0.90 KCNH2 (0.59) KCNH2MC4RCYP3A4CYP2D6CYP2C9
SCHEMBL3346440 0.90 KCNH2 (0.59) KCNH2MC4RCYP3A4CYP2D6CYP2C9
SCHEMBL3346321 0.84 KCNH2 (0.77) KCNH2MC4RCYP3A4CYP2D6CYP2C9
SCHEMBL3350446 0.82 KCNH2 (0.79) KCNH2MC4RCYP3A4CYP2D6CYP2C9
SCHEMBL13365061 0.82 KCNH2 (0.79) KCNH2MC4RCYP3A4CYP2D6CYP2C9
SCHEMBL3353012 0.81 KCNH2 (0.59) KCNH2MC4RCYP3A4CYP2D6CYP2C9
SCHEMBL3346236 0.81 MC4R (0.65) KCNH2MC4RCYP3A4CYP2D6CYP2C9
SCHEMBL13365134 0.79 KCNH2 (0.64) KCNH2MC4RCYP3A4CYP2D6CYP2C9
SCHEMBL13365062 0.78 KCNH2 (0.57) KCNH2MC4RCYP3A4CYP2D6CYP2C9
SCHEMBL3346870 0.78 KCNH2 (0.62) KCNH2MC4RCYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed