SCHEMBL3353012

SCHEMBL3353012

CC[C@H](NC(=O)[C@@H]1CNC[C@H]1c1ccc(C(F)(F)F)cc1)c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.59
KCNA5 P22460 1/20 0.48
GPR88 Q9GZN0 1/20 0.47
KCNQ3 O43525 3/20 0.44
KCNQ2 O43526 3/20 0.44
KCNQ4 P56696 1/20 0.44
KCNQ5 Q9NR82 1/20 0.44
TDP1 Q9NUW8 1/20 0.43
MC4R P32245 1/20 0.43
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
FFAR1 O14842 1/20 0.41
TACR1 P25103 3/20 0.41
SLC6A9 P48067 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3353295 0.87 GPR88 (0.52) KCNH2GPR88KCNQ3KCNQ2TDP1
SCHEMBL3346321 0.86 KCNH2 (0.77) KCNH2KCNQ3KCNQ2KCNQ4KCNQ5
SCHEMBL3346433 0.84 KCNH2 (0.56) KCNH2
SCHEMBL3346531 0.84 GPR88 (0.66) KCNH2KCNA5GPR88KCNQ3KCNQ2
SCHEMBL3346210 0.81 KCNH2 (0.59) KCNH2MC4RCYP3A4CYP2D6CYP2C9
SCHEMBL3416539 0.81 GPR88 (0.45) KCNH2GPR88KCNQ3KCNQ2KCNQ4
SCHEMBL3353261 0.81 GPR88 (0.46) GPR88KCNQ3KCNQ2KCNQ4KCNQ5
SCHEMBL13365061 0.78 KCNH2 (0.79) KCNH2MC4RCYP3A4CYP2D6CYP2C9
SCHEMBL3350446 0.78 KCNH2 (0.79) KCNH2MC4RCYP3A4CYP2D6CYP2C9
SCHEMBL3346364 0.78 KCNH2 (0.68) KCNH2KCNQ3KCNQ2KCNQ4KCNQ5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed