SCHEMBL335390

SCHEMBL335390

Nc1nc2ccc(NC(=O)C(O)C(NC(=O)c3ccc4ccccc4c3)c3ccccc3)cc2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.44
FABP6 P51161 1/20 0.44
PIN1 Q13526 4/20 0.44
ACP1 P24666 1/20 0.41
F9 P00740 2/20 0.41
F7 P08709 2/20 0.41
CTSL P07711 1/20 0.40
CTSK P43235 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
F11 P03951 1/20 0.38
CHEK2 O96017 1/20 0.38
TP53 P04637 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL335500 0.92 F9 (0.44) ABL1FABP6F9F7MEN1
SCHEMBL336367 0.91 MAPT (0.47) ABL1FABP6ACP1F9F7
SCHEMBL335878 0.90 ABL1 (0.43) ABL1FABP6ACP1F9F7
SCHEMBL335948 0.90 ABL1 (0.45) ABL1FABP6ACP1F9F7
SCHEMBL336586 0.89 GRIN1 (0.44) ABL1FABP6ACP1F9F7
SCHEMBL334843 0.89 KDR (0.45) ABL1FABP6F9F7MEN1
SCHEMBL8219489 0.88 F9 (0.43) ABL1FABP6ACP1F9F7
SCHEMBL335576 0.88 ABL1 (0.43) ABL1FABP6ACP1F9F7
SCHEMBL335205 0.87 TYMS (0.42) ABL1FABP6ACP1F9F7
SCHEMBL335420 0.87 NPC1 (0.46) ABL1FABP6F9F7MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8097758-B2 Isoserine derivatives for use as coagulation factor IXa inhibitors SANOFI-AVENTIS (FR) 2012-01-17 US claimed