SCHEMBL3354417

SCHEMBL3354417

N#CC1(Cc2ccc(F)nc2)CCN(C(=O)O)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.40
FPR2 P25090 1/20 0.34
PROKR1 Q8TCW9 1/20 0.34
PRKAA2 P54646 2/20 0.34
C3AR1 Q16581 1/20 0.34
SPR P35270 2/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
CYP2C9 P11712 2/20 0.33
TSHR P16473 2/20 0.33
CYP2D6 P10635 1/20 0.33
VNN1 O95497 1/20 0.33
HIF1A Q16665 1/20 0.32
KDM1A O60341 1/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
P2RX7 Q99572 1/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3355141 0.83 JAK2 (0.49) JAK2JAK1
SCHEMBL2798597 0.83 ALDH1A1 (0.43) ALDH1A1FPR2PROKR1PRKAA2
SCHEMBL5811202 0.79 ALDH1A1 (0.43) ALDH1A1CYP2D6MEN1KMT2A
SCHEMBL18321618 0.78 NPSR1 (0.41) ALDH1A1FPR2PROKR1CYP2D6
SCHEMBL3352880 0.77 KDM1A (0.33) FPR2PROKR1TSHRCYP2D6KDM1A
SCHEMBL23647559 0.72 CYP46A1 (0.44) ALDH1A1JAK2JAK1TSHR
SCHEMBL3116168 0.72 MEN1 (0.53) PRKAA2MEN1KMT2A
SCHEMBL28123143 0.72 CHRM2 (0.46) ALDH1A1TSHRMEN1KMT2A
SCHEMBL22719293 0.71 MGLL (0.43) JAK2JAK1
SCHEMBL18321417 0.71 ESR2 (0.42) FPR2PROKR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010068881-A1 NOVEL BENZODIOXANE AND BENZOXAZINE DERIVATIVES USEFUL AS CC CHEMOKINE RECEPTOR LIGANDS FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-06-17 WO disclosed