SCHEMBL3354842

SCHEMBL3354842

NC(Cc1nc(O)c2cc(-c3ccncc3)ccc2n1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.48
AAK1 Q2M2I8 10/20 0.42
CHEK1 O14757 1/20 0.41
GSK3B P49841 1/20 0.41
MKNK1 Q9BUB5 1/20 0.41
BMP2K Q9NSY1 1/20 0.41
PIK3CA P42336 1/20 0.40
DPP4 P27487 1/20 0.40
DPP8 Q6V1X1 1/20 0.40
MAP4K4 O95819 3/20 0.40
AKT1 P31749 2/20 0.40
CLK2 P49760 2/20 0.40
ROCK1 Q13464 2/20 0.40
DYRK1A Q13627 2/20 0.40
CLK4 Q9HAZ1 2/20 0.40
PRKD3 O94806 1/20 0.40
PRKCG P05129 1/20 0.40
PIM1 P11309 1/20 0.40
PRKACA P17612 1/20 0.40
RPS6KB1 P23443 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3354836 0.79 ROCK2 (0.59) ROCK2AAK1CHEK1GSK3BMKNK1
SCHEMBL3354838 0.79 ROCK2 (0.59) ROCK2AAK1CHEK1GSK3BMKNK1
SCHEMBL17653243 0.72 AAK1 (0.73) AAK1CHEK1GSK3BMKNK1BMP2K
SCHEMBL3355527 0.68 ROCK2 (0.46) ROCK2CHEK1GSK3BMAP4K4ROCK1
SCHEMBL18040189 0.66 GRIN2D (0.67) DPP4
SCHEMBL3496826 0.65 TRIM58 (0.45) PIK3CAMAP4K4
SCHEMBL1157043 0.65 SLC6A4 (0.60) DPP4
SCHEMBL16974250 0.64 PDGFRB (0.49) AAK1CHEK1GSK3BMKNK1BMP2K
Hydrochloric Acid SCHEMBL9322405 0.64 SLC6A4 (0.58) DPP4
Hydrochloric Acid SCHEMBL9322527 0.64 SLC6A4 (0.58) DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010056758-A1 QUINAZOLINE DERIVATIVES AS KINASE INHIBITORS FENG YANGBO (US) 2010-05-20 WO disclosed