SCHEMBL3357892

SCHEMBL3357892

COc1ccc(CNC(O)CCNC(=O)O)cc1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CASR P41180 1/20 0.54
NPC1 O15118 4/20 0.48
RAB9A P51151 3/20 0.47
HPGD P15428 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.46
ALDH1A1 P00352 3/20 0.46
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
ATM Q13315 1/20 0.46
PKM P14618 1/20 0.45
LDHA P00338 1/20 0.45
GAA P10253 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3356473 0.85 SMN1; SMN2 (0.49) NPC1RAB9AHPGDSMN1; SMN2ALDH1A1
SCHEMBL3348575 0.84 ALDH1A1 (0.55) RAB9AHPGDSMN1; SMN2ALDH1A1KMT2A
SCHEMBL3350274 0.83 EPHX2 (0.46) SMN1; SMN2
SCHEMBL5433856 0.81 GAA (0.51) HPGDALDH1A1KMT2AMEN1ATM
SCHEMBL1695235 0.78 NPC1 (0.66) NPC1RAB9AHPGDSMN1; SMN2ALDH1A1
SCHEMBL5435357 0.78 MEN1 (0.48) ALDH1A1KMT2AMEN1TDP1
SCHEMBL19280078 0.78 MEN1 (0.62) NPC1RAB9AHPGDSMN1; SMN2ALDH1A1
SCHEMBL3351114 0.78 KCNH2 (0.45) ALDH1A1KMT2AMEN1
SCHEMBL22028845 0.77 ALDH1A1 (0.50) CASRNPC1RAB9AHPGDSMN1; SMN2
SCHEMBL11728101 0.77 ALDH1A1 (0.57) NPC1SMN1; SMN2ALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7727997-B2 N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives ELAN PHARMACEUTICALS, INC. (US) 2010-06-01 US disclosed
US-20070213316-A1 Compounds that are effective inhibitors of beta-secretase; inhibitors of beta-secretase-mediated cleavage of amyloid precursor proteins; effective inhibitors of A beta production, and/or are effective to reduce amyloid beta deposits or plaques; treatment of disorders such as Alzheimer's Disease ELAN PHARMACEUTICALS, INC. 2007-09-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070213316-A1 Compounds that are effective inhibitors of beta-secretase; inhibitors of beta-secretase-mediated cleavage of amyloid precursor proteins; effective inhibitors of A beta production, and/or are effective to reduce amyloid beta deposits or plaques; treatment of disorders such as Alzheimer's Disease BACE1, BACE2, APP CASR 2012/4885NPC1 593/4885RAB9A 874/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.