SCHEMBL3348575

SCHEMBL3348575

COc1cccc(CNC(O)CCNC(=O)O)c1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.55
HTT P42858 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
MMP13 P45452 3/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
APEX1 P27695 1/20 0.49
BCHE P06276 1/20 0.48
LMNA P02545 1/20 0.48
MTNR1A P48039 2/20 0.48
MTNR1B P49286 2/20 0.48
RAB9A P51151 1/20 0.48
POLB P06746 1/20 0.48
HPGD P15428 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3351538 0.84 MAPK14 (0.53) MMP13
SCHEMBL3357892 0.84 CASR (0.54) ALDH1A1SMN1; SMN2MEN1KMT2ARAB9A
SCHEMBL5065712 0.82 ALDH1A1 (0.51) ALDH1A1HTTSMN1; SMN2MMP13MEN1
SCHEMBL2931410 0.81 MMP13 (0.70) ALDH1A1HTTSMN1; SMN2MMP13MEN1
SCHEMBL5433856 0.79 GAA (0.51) ALDH1A1MEN1KMT2AMTNR1AMTNR1B
SCHEMBL2205978 0.78 MTNR1A (0.65) ALDH1A1HTTSMN1; SMN2MEN1KMT2A
SCHEMBL3355242 0.78 BCHE (0.49) MEN1KMT2ABCHELMNARAB9A
SCHEMBL5433128 0.77 CASR (0.50) ALDH1A1HTTSMN1; SMN2MMP13MEN1
SCHEMBL5435357 0.77 MEN1 (0.48) ALDH1A1MEN1KMT2A
SCHEMBL5069135 0.76 MTNR1A (0.62) ALDH1A1HTTMEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7727997-B2 N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives ELAN PHARMACEUTICALS, INC. (US) 2010-06-01 US disclosed
US-20070213316-A1 Compounds that are effective inhibitors of beta-secretase; inhibitors of beta-secretase-mediated cleavage of amyloid precursor proteins; effective inhibitors of A beta production, and/or are effective to reduce amyloid beta deposits or plaques; treatment of disorders such as Alzheimer's Disease ELAN PHARMACEUTICALS, INC. 2007-09-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070213316-A1 Compounds that are effective inhibitors of beta-secretase; inhibitors of beta-secretase-mediated cleavage of amyloid precursor proteins; effective inhibitors of A beta production, and/or are effective to reduce amyloid beta deposits or plaques; treatment of disorders such as Alzheimer's Disease BACE1, BACE2, APP ALDH1A1 2133/4885HTT 493/4885SMN1; SMN2 1298/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.