SCHEMBL3358245

SCHEMBL3358245

COc1nccc2cc(-c3ccccc3)ncc12

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 10/20 0.59
IDO1 P14902 9/20 0.59
NPC1 O15118 4/20 0.54
RAB9A P51151 3/20 0.54
SQOR Q9Y6N5 3/20 0.45
MAPT P10636 2/20 0.44
MEN1 O00255 1/20 0.44
TSHR P16473 1/20 0.44
KMT2A Q03164 1/20 0.44
ATM Q13315 1/20 0.44
ALDH1A1 P00352 1/20 0.43
GLA P06280 1/20 0.43
GAA P10253 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30081970 0.77 TDO2 (0.69) TDO2IDO1NPC1RAB9AMAPT
SCHEMBL22715639 0.74 NPC1 (0.47) NPC1RAB9AMAPTMEN1TSHR
SCHEMBL29472095 0.74 NPC1 (0.47) NPC1RAB9AMAPTMEN1TSHR
SCHEMBL1043405 0.74 SQOR (0.47) TDO2IDO1NPC1RAB9ASQOR
SCHEMBL22715444 0.73 MAPT (0.43) TDO2IDO1NPC1RAB9AMAPT
SCHEMBL24622584 0.73 MAPK10 (0.59) TDO2IDO1NPC1RAB9AMAPT
SCHEMBL8272283 0.72 SQOR (0.60) TDO2IDO1NPC1RAB9ASQOR
SCHEMBL3318438 0.71 NPC1 (0.69) TDO2IDO1NPC1RAB9AMAPT
SCHEMBL2231183 0.71 CYP2A6 (0.55) NPC1RAB9AMAPTTSHRALDH1A1
SCHEMBL30223171 0.71 CYP2A6 (0.55) NPC1RAB9AMAPTTSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2238137-A1 COMPOUNDS AND COMPOSITIONS AS KINASE INHIBITORS IRM LLC (BM) 2010-10-13 EP disclosed
WO-2009097287-A1 COMPOUNDS AND COMPOSITIONS AS KINASE INHIBITORS IRM LLC (BM) 2009-08-06 WO disclosed