SCHEMBL3360284

SCHEMBL3360284

O=c1[nH]c2cccc(Cl)c2c(F)c1O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 3/20 0.60
GRIN3B O60391 3/20 0.60
GRIN1 Q05586 3/20 0.60
GRIN2A Q12879 3/20 0.60
GRIN2B Q13224 3/20 0.60
GRIN2C Q14957 3/20 0.60
GRIN3A Q8TCU5 3/20 0.60
DAO P14920 3/20 0.50
ERCC5 P28715 1/20 0.49
FEN1 P39748 1/20 0.49
CHEK1 O14757 1/20 0.47
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
IDE P14735 1/20 0.44
MPI P34949 1/20 0.44
CACNA1B Q00975 1/20 0.44
APBA1 Q02410 1/20 0.44
DDO Q99489 2/20 0.42
PBRM1 Q86U86 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3422204 0.81 DAO (0.49) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL3359927 0.79 GRIN2D (0.45) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL3422531 0.79 DAO (0.51) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL3395242 0.78 FASN (0.42) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL3426211 0.76 DAO (0.55) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL3426119 0.75 DAO (0.41) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL3363824 0.75 DAO (0.46) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL9393158 0.75 DAO (0.66) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL27805830 0.75 GPR17 (0.58) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL17942038 0.73 KDM4E (0.69) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010058314-A1 HYDROXYQUINOLIN-2(1H)-ONES AND DERIVATIVES THEREOF PFIZER INC. (US) 2010-05-27 WO claimed
WO-2010058314-A1 HYDROXYQUINOLIN-2(1H)-ONES AND DERIVATIVES THEREOF PFIZER INC. (US) 2010-05-27 WO disclosed