SCHEMBL3360583

SCHEMBL3360583

Cc1nc(CCC(=O)c2ccc(Cl)c(Cl)c2)no1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
MAPT P10636 2/20 0.40
NPC1 O15118 1/20 0.40
POLB P06746 1/20 0.40
RAB9A P51151 1/20 0.40
KMO O15229 3/20 0.40
MGAM O43451 1/20 0.39
AMY1A P0DUB6 1/20 0.39
GAA P10253 1/20 0.39
SI P14410 1/20 0.39
MGAM2 Q2M2H8 1/20 0.39
HDAC4 P56524 3/20 0.39
HDAC1 Q13547 3/20 0.39
HDAC7 Q8WUI4 3/20 0.39
HDAC11 Q96DB2 3/20 0.39
HDAC8 Q9BY41 3/20 0.39
HDAC6 Q9UBN7 3/20 0.39
HDAC9 Q9UKV0 3/20 0.39
HDAC5 Q9UQL6 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12327069 0.84 MEN1 (0.37) MEN1KMT2AMAPTNPC1POLB
SCHEMBL7974742 0.79 DRD4 (0.43) MEN1KMT2AMAPTNPC1POLB
SCHEMBL2433489 0.79 DRD4 (0.43) MEN1KMT2AMAPTNPC1POLB
SCHEMBL2431451 0.79 MEN1 (0.42) MEN1KMT2AMAPTNPC1POLB
SCHEMBL3363237 0.72 MGAM (0.45) MEN1KMT2ANPC1RAB9AKMO
SCHEMBL2433048 0.70 ALDH1A1 (0.43) KMOMGAMAMY1AGAASI
SCHEMBL634176 0.70 HSD17B3 (0.55) MEN1KMT2ANPC1RAB9AKMO
SCHEMBL9337894 0.69 THRA (0.59) KMOHDAC4HDAC1HDAC7HDAC11
SCHEMBL14166820 0.69 TP53 (0.41) POLBRAB9AALDH1A1
SCHEMBL2435064 0.69 KDM4E (0.57) KMOHDAC4HDAC1HDAC7HDAC11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010011302-A1 CERTAIN KYNURENINE-3-MONOOXYGENASE INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF USE THEREOF CHDI, INC. (US) 2010-01-28 WO claimed