SCHEMBL3363097

SCHEMBL3363097

CC(C)NC(=O)Oc1cn(S(=O)(=O)c2ccc(C(C)(C)C)cc2)c2ccc(Cl)cc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 7/20 0.42
FLT1 P17948 1/20 0.41
FLT4 P35916 1/20 0.41
KDR P35968 1/20 0.41
EPHX2 P34913 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
DRD2 P14416 1/20 0.39
SLC6A2 P23975 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
SLC6A4 P31645 1/20 0.39
HTR7 P34969 1/20 0.39
HRH1 P35367 1/20 0.39
ADRA1B P35368 1/20 0.39
SLC6A3 Q01959 1/20 0.39
KCNH2 Q12809 1/20 0.39
ACLY P53396 1/20 0.38
NR1I2 O75469 2/20 0.38
HSD17B2 P37059 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3367219 0.86 MEN1 (0.45) HTR6FLT1FLT4KDRCYP3A4
SCHEMBL3141520 0.85 FLT1 (0.47) HTR6FLT1FLT4KDREPHX2
SCHEMBL3366631 0.85 FLT1 (0.43) HTR6FLT1FLT4KDREPHX2
SCHEMBL3362365 0.85 HTR6 (0.42) HTR6FLT1FLT4KDRCYP3A4
SCHEMBL3361493 0.77 PPARG (0.42) HTR6FLT1FLT4KDRCYP3A4
SCHEMBL3132165 0.76 AKR1C3 (0.50) HTR6FLT1FLT4KDRACLY
SCHEMBL3133901 0.76 PLK1 (0.55) HTR6FLT1FLT4KDREPHX2
SCHEMBL3362896 0.76 HTR6 (0.44) HTR6CYP3A4CYP2D6DRD2SLC6A2
SCHEMBL3137579 0.75 FLT1 (0.46) HTR6FLT1FLT4KDREPHX2
SCHEMBL27713331 0.74 HTR6 (0.48) HTR6MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2118060-B1 1-BENZENESULFONYL-1H-INDOLE DERIVATIVES AS INHIBITORS OF CCR9 ACTIVITY NOVARTIS AG (CH) 2010-10-06 EP claimed