SCHEMBL3365084

SCHEMBL3365084

COc1cc(OC)c2c(CN)ncc(C(=O)N(C)C(C)c3ccccc3)c2c1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 12/20 0.57
EGLN1 Q9GZT9 1/20 0.40
RPS6KB1 P23443 5/20 0.37
AURKA O14965 4/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3366032 0.99 DPP4 (0.58) DPP4EGLN1RPS6KB1AURKAKDM4E
SCHEMBL3363088 0.84 DPP4 (0.41) DPP4EGLN1RPS6KB1AURKAKDM4E
SCHEMBL3363889 0.83 DPP4 (0.59) DPP4
SCHEMBL3361560 0.79 DPP4 (0.74) DPP4
SCHEMBL3361355 0.79 DPP4 (0.55) DPP4KDM4EALDH1A1
Hydrochloric Acid SCHEMBL3365053 0.76 DPP4 (0.55) DPP4KDM4EALDH1A1
SCHEMBL3363205 0.76 DPP4 (0.56) DPP4
SCHEMBL3363200 0.75 DPP4 (0.55) DPP4RPS6KB1ALDH1A1
Hydrochloric Acid SCHEMBL3366027 0.75 DPP4 (0.56) DPP4
Hydrochloric Acid SCHEMBL3366022 0.75 DPP4 (0.55) DPP4RPS6KB1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US claimed
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US disclosed