SCHEMBL3363200

SCHEMBL3363200

COc1cc(OC)c2c(CN)ncc(C(=O)NC(C)c3cccnc3)c2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 5/20 0.55
ROCK1 Q13464 11/20 0.43
PRKACA P17612 4/20 0.43
GSK3A P49840 4/20 0.43
GSK3B P49841 4/20 0.43
PRKX P51817 3/20 0.43
PRKCG P05129 3/20 0.43
RPS6KB1 P23443 3/20 0.43
MAPK1 P28482 3/20 0.43
RPS6KA3 P51812 3/20 0.43
PRKCD Q05655 3/20 0.43
PRKG1 Q13976 3/20 0.43
PKN2 Q16513 3/20 0.43
CLK4 Q9HAZ1 3/20 0.43
SGK2 Q9HBY8 3/20 0.43
AKT3 Q9Y243 3/20 0.43
CDK2 P24941 2/20 0.43
MARK3 P27448 2/20 0.43
AKT1 P31749 2/20 0.43
CLK2 P49760 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3366022 0.99 DPP4 (0.55) DPP4ROCK1PRKACAGSK3AGSK3B
SCHEMBL3363205 0.76 DPP4 (0.56) DPP4MAPK1HPGD
SCHEMBL3365084 0.75 DPP4 (0.57) DPP4RPS6KB1ALDH1A1
Hydrochloric Acid SCHEMBL3366027 0.75 DPP4 (0.56) DPP4MAPK1HPGD
SCHEMBL3361560 0.75 DPP4 (0.74) DPP4
SCHEMBL7716544 0.75 DPP4 (0.65) DPP4MAPK1
Hydrochloric Acid SCHEMBL3366032 0.75 DPP4 (0.58) DPP4RPS6KB1ALDH1A1
SCHEMBL3362414 0.74 DPP4 (0.61) DPP4ROCK1ROCK2ALDH1A1HPGD
Hydrochloric Acid SCHEMBL3361903 0.74 DPP4 (0.62) DPP4ROCK1ROCK2ALDH1A1HPGD
SCHEMBL3362219 0.70 GAA (0.49) DPP4ROCK1MAPK1ROCK2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US claimed
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US disclosed