SCHEMBL3365216

SCHEMBL3365216

COc1ccc(CNC(=O)Cc2cnc(CN)c3cc(OC)c(OC)cc23)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 9/20 0.58
NPC1 O15118 2/20 0.49
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
HTT P42858 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HSD17B10 Q99714 1/20 0.47
ERCC1 P07992 1/20 0.46
ERCC4 Q92889 1/20 0.46
ALDH1A1 P00352 1/20 0.45
POLB P06746 1/20 0.45
RAB9A P51151 1/20 0.45
MAPT P10636 1/20 0.45
BCHE P06276 1/20 0.45
ACHE P22303 1/20 0.45
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
PDE10A Q9Y233 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3361314 0.84 NPC1 (0.44) DPP4NPC1CA12CA1CA2
SCHEMBL3361885 0.84 DPP4 (0.67) DPP4HSD17B10ALDH1A1POLBRAB9A
Hydrochloric Acid SCHEMBL3364779 0.83 DPP4 (0.68) DPP4ALDH1A1POLBRAB9ABCHE
SCHEMBL3360544 0.81 DPP4 (0.61) DPP4PDE10A
Hydrochloric Acid SCHEMBL3369616 0.81 DPP4 (0.62) DPP4PDE10A
SCHEMBL8289766 0.80 DPP4 (0.59) DPP4SMN1; SMN2ALDH1A1
SCHEMBL7723652 0.78 DPP4 (0.73) DPP4HSD17B10PDE10A
SCHEMBL13792321 0.74 DPP4 (1.00) DPP4PDE10A
SCHEMBL3362414 0.73 DPP4 (0.61) DPP4SMN1; SMN2HSD17B10ALDH1A1POLB
Hydrochloric Acid SCHEMBL29356163 0.73 DPP4 (1.00) DPP4PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US claimed
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US disclosed
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US disclosed
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US disclosed