SCHEMBL3361885

SCHEMBL3361885

COc1ccc(CNC(=O)c2cnc(CN)c3cc(OC)c(OC)cc23)cc1

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 9/20 0.67
PDE10A Q9Y233 1/20 0.56
ALDH1A1 P00352 3/20 0.49
HPGD P15428 3/20 0.49
KDM4E B2RXH2 2/20 0.49
PKM P14618 1/20 0.49
KLKB1 P03952 1/20 0.49
RAB9A P51151 1/20 0.48
CYP1A2 P05177 1/20 0.48
POLB P06746 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
ATM Q13315 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
TSHR P16473 1/20 0.48
BCHE P06276 1/20 0.48
ACHE P22303 1/20 0.48
HSD17B10 Q99714 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3364779 0.99 DPP4 (0.68) DPP4PDE10AALDH1A1HPGDKDM4E
SCHEMBL3362414 0.86 DPP4 (0.61) DPP4PDE10AALDH1A1HPGDKDM4E
Hydrochloric Acid SCHEMBL3361903 0.85 DPP4 (0.62) DPP4PDE10AALDH1A1HPGDKDM4E
SCHEMBL3365216 0.84 DPP4 (0.58) DPP4PDE10AALDH1A1RAB9APOLB
SCHEMBL3365143 0.84 PDE10A (0.51) DPP4PDE10AALDH1A1HPGDKDM4E
SCHEMBL7716787 0.81 DPP4 (1.00) DPP4PDE10AALDH1A1HPGDPOLB
SCHEMBL3360594 0.76 DPP4 (0.71) DPP4
SCHEMBL3365202 0.74 DPP4 (0.44) DPP4PDE10AALDH1A1HPGDKDM4E
SCHEMBL17581348 0.73 HPGD (0.53) ALDH1A1HPGDKDM4EPKMKLKB1
SCHEMBL3361845 0.72 DPP4 (1.00) DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US claimed
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US disclosed
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US disclosed
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US disclosed