SCHEMBL3365929

SCHEMBL3365929

O=C(O)Oc1sc2cc(O)c(O)c([N+](=O)[O-])c2c1Cl

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
COMT P21964 12/20 0.46
CDK2 P24941 2/20 0.39
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33
GRIN2C Q14957 1/20 0.33
GRIN3A Q8TCU5 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
TTR P02766 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1608964 0.80 COMT (0.46) COMTCDK2ALDH1A1CYP1A2CYP2D6
SCHEMBL3365763 0.80 COMT (0.65) COMTCDK2ALDH1A1CYP1A2CYP2D6
SCHEMBL1608806 0.71 HPGD (0.58) COMTALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL1608929 0.70 CDK2 (0.44) COMTCDK2
SCHEMBL3364327 0.68 COMT (0.47) COMTCDK2
SCHEMBL3364756 0.67 COMT (0.61) COMTCDK2
SCHEMBL3363596 0.66 COMT (0.60) COMTCDK2
SCHEMBL3362922 0.65 COMT (0.55) COMTCDK2CYP1A2CYP2D6CYP2C19
SCHEMBL1608186 0.64 COMT (0.73) COMTCDK2ALDH1A1CYP1A2CYP2D6
SCHEMBL11295224 0.63 GRIN2D (0.50) COMTCDK2GRIN2DGRIN3BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910325-B1 NEW PHARMACEUTICAL COMPOUNDS ORION CORP (FI) 2010-10-06 EP claimed