SCHEMBL3366814

SCHEMBL3366814

CCC(C)(C)c1ccc(CS(=O)(=O)N2CCCC2c2nnc(-c3ccc(Cl)cc3)o2)cc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.41
HPGD P15428 4/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
MAPT P10636 2/20 0.41
POLB P06746 1/20 0.40
CYP2D6 P10635 1/20 0.40
ALDH1A1 P00352 2/20 0.40
ALOX15B O15296 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.38
LMNA P02545 1/20 0.38
HSD11B1 P28845 1/20 0.37
S1PR4 O95977 2/20 0.35
S1PR1 P21453 2/20 0.35
S1PR5 Q9H228 2/20 0.35
S1PR3 Q99500 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3366972 0.91 USP30 (0.41) KDM4EHPGDCYP3A4CYP2C9CYP2C19
SCHEMBL3366848 0.90 ALDH1A1 (0.48) KDM4EHPGDCYP3A4CYP2C9CYP2C19
SCHEMBL3370219 0.85 KDM4E (0.49) KDM4EHPGDCYP3A4CYP2C9CYP2C19
SCHEMBL3370504 0.84 CYP2C19 (0.43) KDM4EHPGDCYP3A4CYP2C9CYP2C19
SCHEMBL3367339 0.79 CYP2C19 (0.43) KDM4ECYP2C19MAPTALDH1A1SMN1; SMN2
SCHEMBL3367261 0.77 SMN1; SMN2 (0.41) KDM4EHPGDCYP3A4CYP2C9CYP2C19
SCHEMBL3370139 0.75 USP30 (0.43) KDM4EHPGDCYP3A4CYP2C9CYP2C19
SCHEMBL6069033 0.75 MAPT (0.42) MAPTPOLBALDH1A1ALOX15BSMN1; SMN2
SCHEMBL3366078 0.75 HCRTR1 (0.46) KDM4ECYP2C19MAPTPOLBALDH1A1
SCHEMBL3368142 0.75 CYP2C19 (0.44) KDM4EHPGDCYP2C19POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1532141-B1 2-PYRROLIDIN-2-YL- [1,3,4]-OXADIAZOLE DERIVATIVES AND THE USE OF THE SAME AS ANTIDEPRESSANTS GRUENENTHAL GMBH (DE) 2010-10-13 EP disclosed