SCHEMBL3368142

SCHEMBL3368142

O=S(=O)(Cc1ccccc1)N1CCCC1c1nnc(-c2ccncc2)o1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.44
USP30 Q70CQ3 1/20 0.43
FKBP1A P62942 2/20 0.41
ALDH1A1 P00352 3/20 0.41
HCRTR1 O43613 1/20 0.41
HCRTR2 O43614 1/20 0.41
DPP4 P27487 1/20 0.41
POLB P06746 2/20 0.41
KDM4E B2RXH2 1/20 0.41
HPGD P15428 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
ATAD2 Q6PL18 1/20 0.40
GSK3B P49841 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.40
GSK3A P49840 1/20 0.40
CCR4 P51679 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3370504 0.90 CYP2C19 (0.43) CYP2C19ALDH1A1POLBKDM4EHPGD
SCHEMBL3367339 0.90 CYP2C19 (0.43) CYP2C19USP30ALDH1A1HCRTR1HCRTR2
SCHEMBL3364395 0.89 ALDH1A1 (0.49) CYP2C19USP30FKBP1AALDH1A1NPC1
SCHEMBL3366078 0.87 HCRTR1 (0.46) CYP2C19FKBP1AALDH1A1HCRTR1HCRTR2
SCHEMBL3368542 0.87 GPR142 (0.48) CYP2C19USP30ALDH1A1HCRTR1HCRTR2
SCHEMBL3370281 0.86 MAPT (0.44) CYP2C19ALDH1A1POLBKDM4ENPC1
SCHEMBL3370219 0.85 KDM4E (0.49) CYP2C19USP30FKBP1AALDH1A1DPP4
SCHEMBL3370356 0.84 ALDH1A1 (0.51) CYP2C19FKBP1AALDH1A1HCRTR1HCRTR2
SCHEMBL3366848 0.83 ALDH1A1 (0.48) CYP2C19FKBP1AALDH1A1POLBKDM4E
SCHEMBL3370780 0.82 CYP2C19 (0.41) CYP2C19USP30ALDH1A1HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1532141-B1 2-PYRROLIDIN-2-YL- [1,3,4]-OXADIAZOLE DERIVATIVES AND THE USE OF THE SAME AS ANTIDEPRESSANTS GRUENENTHAL GMBH (DE) 2010-10-13 EP disclosed