SCHEMBL3371272

SCHEMBL3371272

Cc1cc(SC/C=C(\C#CC(C)(C)O)c2ccc(-c3ccccc3)cc2)ccc1O

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 3/20 0.33
ESR1 P03372 4/20 0.33
ESR2 Q92731 4/20 0.33
HSD17B1 P14061 3/20 0.33
HSD17B2 P37059 3/20 0.33
PPARA Q07869 1/20 0.31
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C19 P33261 1/20 0.30
ALPL P05186 1/20 0.30
GAA P10253 1/20 0.30
ALPG P10696 1/20 0.30
PLAA Q9Y263 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3372729 0.85 PPARD (0.34) PPARDESR1ESR2HSD17B1HSD17B2
SCHEMBL3032424 0.84 PPARD (0.55) PPARDPPARA
SCHEMBL3032421 0.84 PPARD (0.55) PPARDPPARA
SCHEMBL3032217 0.81 PPARA (0.43) PPARDPPARA
SCHEMBL3034484 0.81 PPARA (0.43) PPARDPPARA
SCHEMBL3373878 0.79 PPARD (0.48) PPARDPPARACYP3A4ALPG
SCHEMBL3375669 0.76 PPARD (0.44) PPARDPPARACYP3A4CYP2D6CYP2C19
SCHEMBL3372723 0.74 PPARD (0.36) PPARDPPARAGAA
SCHEMBL3372726 0.74 PPARD (0.36) PPARDPPARAGAA
SCHEMBL3375341 0.72 PPARD (0.44) PPARDCYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745002-B1 NOVEL COMPOUNDS, THEIR PREPARATION AND USE HIGH POINT PHARMACEUTICALS LLC (US) 2010-11-03 EP claimed