SCHEMBL3371398

SCHEMBL3371398

COc1ccc2nccc(C(CO)[C@]3(O)CC[C@@H](N)CC3)c2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 9/20 0.44
KDM4E B2RXH2 6/20 0.44
ALDH1A1 P00352 5/20 0.44
HSD17B10 Q99714 5/20 0.44
ADRA2A P08913 4/20 0.44
SLC6A4 P31645 4/20 0.44
OPRM1 P35372 4/20 0.44
KCNH2 Q12809 4/20 0.44
HPGD P15428 3/20 0.44
CYP3A4 P08684 3/20 0.44
TSHR P16473 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
SLC6A3 Q01959 2/20 0.44
CHRM2 P08172 1/20 0.44
SLC22A12 Q96S37 1/20 0.42
SLC22A1 O15245 3/20 0.42
ABCB11 O95342 3/20 0.42
ABCB1 P08183 3/20 0.42
SCN1A P35498 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3371400 0.79 ROCK2 (0.47) CYP2D6KDM4EALDH1A1HSD17B10ADRA2A
SCHEMBL7017484 0.78 CYP2D6 (0.48) CYP2D6KDM4EALDH1A1HSD17B10ADRA2A
SCHEMBL3686476 0.74 MTNR1A (0.51) KDM4EKCNH2SLC22A12LMNA
SCHEMBL3377631 0.74 CYP2D6 (0.46) CYP2D6KDM4EALDH1A1HSD17B10ADRA2A
SCHEMBL3377628 0.74 CYP2D6 (0.46) CYP2D6KDM4EALDH1A1HSD17B10ADRA2A
SCHEMBL4269291 0.74 SLC2A1 (0.63) CYP2D6KDM4EALDH1A1HSD17B10ADRA2A
SCHEMBL5256391 0.74 SLC2A1 (0.63) CYP2D6KDM4EALDH1A1HSD17B10ADRA2A
SCHEMBL5256396 0.74 SLC2A1 (0.63) CYP2D6KDM4EALDH1A1HSD17B10ADRA2A
Hydrochloric Acid SCHEMBL5411589 0.73 SLC2A1 (0.62) CYP2D6KDM4EALDH1A1HSD17B10ADRA2A
Oxalic Acid SCHEMBL5253830 0.70 SLC2A1 (0.64) KCNH2SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1987040-B1 ETHANOL OR 1,2-ETHANEDIOL CYCLOHEXYL ANTIBIOTIC DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-11-10 EP disclosed