SCHEMBL3371941

SCHEMBL3371941

Oc1cccc2cc(Br)sc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.53
MEN1 O00255 3/20 0.39
ALDH1A1 P00352 3/20 0.39
KMT2A Q03164 3/20 0.39
DNMT1 P26358 1/20 0.39
CACNA1B Q00975 1/20 0.39
APBA1 Q02410 1/20 0.39
MCL1 Q07820 1/20 0.39
APOBEC3G Q9HC16 1/20 0.39
CYP1A2 P05177 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HDAC8 Q9BY41 3/20 0.35
HDAC3 O15379 2/20 0.35
HDAC4 P56524 2/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC7 Q8WUI4 2/20 0.35
HDAC2 Q92769 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29379963 0.78 CA2 (0.56) CA2MEN1ALDH1A1KMT2ADNMT1
SCHEMBL23500126 0.78 PSMB8 (0.38) CA2MEN1ALDH1A1KMT2AMCL1
SCHEMBL28134157 0.78 CA2 (0.56) CA2MEN1ALDH1A1KMT2ADNMT1
SCHEMBL4806043 0.77 CA2 (0.55) CA2MEN1ALDH1A1KMT2ADNMT1
SCHEMBL31125053 0.75 HDAC3 (0.54) CYP1A2HDAC8HDAC3HDAC4HDAC1
SCHEMBL23220879 0.75 HDAC3 (0.54) CYP1A2HDAC8HDAC3HDAC4HDAC1
SCHEMBL30250636 0.74 CYP2A6 (0.31)
SCHEMBL14780084 0.74 CYP2A6 (0.31)
SCHEMBL6229401 0.73 NR4A1 (0.44) CA2MEN1ALDH1A1KMT2AHDAC8
SCHEMBL28660108 0.72 MGLL (0.53) CA2MEN1ALDH1A1KMT2ADNMT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537091-B1 NOVEL 2-ARYLTHIAZOLE COMPOUNDS AS PPARALPHA AND PPARGAMMA AGONISTS HOFFMANN LA ROCHE (CH) 2010-10-06 EP disclosed