SCHEMBL3374766

SCHEMBL3374766

Cc1cc(C(F)(F)F)ccc1N1C(=O)c2cccc(O)c2C1=O

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 3/20 0.51
ANPEP P15144 2/20 0.51
TYMS P04818 2/20 0.47
ESR1 P03372 1/20 0.45
ESR2 Q92731 1/20 0.45
GRM1 Q13255 6/20 0.43
GRM4 Q14833 6/20 0.43
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
POLB P06746 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3374587 0.90 ANPEP (0.46) DPP4ANPEPTYMSESR1ESR2
SCHEMBL3377225 0.90 ANPEP (0.46) DPP4ANPEPTYMSESR1ESR2
SCHEMBL3373257 0.83 LMNA (0.47) DPP4ANPEPTYMSESR1ESR2
SCHEMBL3374723 0.80 LMNA (0.47) DPP4TYMSGRM1GRM4LMNA
SCHEMBL3373539 0.80 ANPEP (0.54) DPP4ANPEPTYMS
SCHEMBL3378400 0.79 LMNA (0.48) DPP4TYMSESR1ESR2GRM1
SCHEMBL3377243 0.77 LMNA (0.47) DPP4GRM1GRM4LMNASMN1; SMN2
SCHEMBL2916208 0.76 GRM1 (0.52) GRM1GRM4LMNASMN1; SMN2
SCHEMBL5429466 0.75 GRM1 (0.51) GRM1GRM4LMNASMN1; SMN2
SCHEMBL5418153 0.75 LMNA (0.42) DPP4TYMSESR1ESR2GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1517886-B1 NOVEL PHTHALAMIDE DERIVATIVES BAYER CROPSCIENCE AG (DE) 2010-11-10 EP disclosed
US-7132455-B2 Phthalamide derivatives BAYER CROPSCIENCE AG (DE) 2006-11-07 US disclosed
US-20060035967-A1 Novel phthalamide derivatives BAYER INTELLECTUAL PROPERTY GMBH (DE) 2006-02-16 US disclosed
EP-1517886-A1 NOVEL PHTHALAMIDE DERIVATIVES Bayer CropScience AG (DE) 2005-03-30 EP disclosed
WO-2004000796-A1 NOVEL PHTHALAMIDE DERIVATIVES BAYER CROPSCIENCE AG (DE) 2003-12-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060035967-A1 Novel phthalamide derivatives HDAC1, HDAC2, CRY1 DPP4 1795/4885ANPEP 3368/4885TYMS 4744/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.