SCHEMBL3375707

SCHEMBL3375707

CC(C)(C)OC(=O)NC(=O)c1c(Cl)cccc1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 2/20 0.46
TAS1R3 Q7RTX0 2/20 0.44
TAS1R1 Q7RTX1 2/20 0.44
TAS1R2 Q8TE23 2/20 0.44
MAPT P10636 2/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
PPIA P62937 1/20 0.43
POLB P06746 2/20 0.43
GAA P10253 2/20 0.43
ALDH1A1 P00352 2/20 0.42
JAK2 O60674 2/20 0.42
JAK1 P23458 2/20 0.42
TYK2 P29597 2/20 0.42
HPGD P15428 1/20 0.42
CYP3A4 P08684 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11987241 0.89 GAA (0.56) MAPTPPIAPOLBGAAJAK2
SCHEMBL25051908 0.78 LMNA (0.54) LCKTAS1R3TAS1R1TAS1R2MAPT
SCHEMBL25051949 0.77 GAA (0.57) MAPTPOLBGAAJAK2JAK1
SCHEMBL3986856 0.76 PBRM1 (0.49) LCKALDH1A1MEN1KMT2A
SCHEMBL31135421 0.76 REN (0.36) LCKPOLBGAAHPGDMEN1
SCHEMBL21358871 0.75 ITGB1 (0.48)
SCHEMBL21358869 0.75 ITGB1 (0.48)
SCHEMBL406889 0.75 MAPK1 (0.45) MAPTPOLBGAAHPGDMEN1
SCHEMBL21484075 0.75 POLB (0.59) POLBGAAHPGDCYP3A4MEN1
SCHEMBL15600324 0.75 GAA (0.56) LCKMAPTPOLBGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029549-B1 PHENYL-PYRAZOLE DERIVATIVES AS NON-STEROIDAL GLUCOCORICOID RECEPTOR LIGANDS GLAXO GROUP LTD (GB) 2010-11-10 EP disclosed