SCHEMBL3378673

SCHEMBL3378673

BrN(Br)CCc1c[nH]c2ccccc12

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.70
HTR1A P08908 5/20 0.70
HTR2C P28335 4/20 0.70
HTR2B P41595 3/20 0.70
HTR6 P50406 4/20 0.66
TRPM8 Q7Z2W7 1/20 0.62
TRPV1 Q8NER1 1/20 0.62
SLC6A4 P31645 2/20 0.61
CYP3A4 P08684 3/20 0.61
HTR1D P28221 2/20 0.61
HTR1B P28222 2/20 0.61
HTR7 P34969 2/20 0.61
CYP2D6 P10635 2/20 0.61
MPO P05164 1/20 0.61
CYP1A2 P05177 1/20 0.61
CYP2A6 P11509 1/20 0.61
NFKB1 P19838 1/20 0.61
CTSK P43235 1/20 0.61
CYP2A13 Q16696 1/20 0.61
TAAR1 Q96RJ0 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9393120 0.98 HTR2A (0.68) HTR2AHTR1AHTR2CHTR2BHTR6
SCHEMBL3380053 0.86 HTR2A (0.66) HTR2AHTR1AHTR2CHTR2BHTR6
SCHEMBL4985934 0.82 HTR2A (0.77) HTR2AHTR1AHTR2CHTR2BHTR6
SCHEMBL3378323 0.82 HTR2A (0.70) HTR2AHTR1AHTR2CHTR2BHTR6
SCHEMBL6933897 0.82 HTR2A (0.70) HTR2AHTR1AHTR2CHTR2BHTR6
SCHEMBL30896267 0.82 HTR2A (0.81) HTR2AHTR1AHTR2CHTR2BHTR6
N,N-Dimethyltryptamine SCHEMBL335710 0.82 HTR2A (1.00) HTR2AHTR1AHTR2CHTR2BHTR6
N,N-Dimethyltryptamine SCHEMBL29350959 0.82 HTR2A (1.00) HTR2AHTR1AHTR2CHTR2BHTR6
SCHEMBL6602711 0.82 HTR2A (0.70) HTR2AHTR1AHTR2CHTR2BHTR6
N,N-Dimethyltryptamine SCHEMBL27221709 0.82 HTR2A (1.00) HTR2AHTR1AHTR2CHTR2BHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010017405-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT OF PAIN HELLER ADAM (US) 2010-02-11 WO claimed
WO-2010017405-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT OF PAIN HELLER ADAM (US) 2010-02-11 WO disclosed