SCHEMBL3380733

SCHEMBL3380733

CN1CCc2ccc(NC(=O)C(CCC(=O)N(C)C)NC(=O)Oc3ccc(Cl)s3)cc2CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 1/20 0.37
F10 P00742 10/20 0.35
ROCK2 O75116 1/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
CA9 Q16790 1/20 0.33
DRD2 P14416 1/20 0.33
HTR2C P28335 1/20 0.33
DRD3 P35462 1/20 0.33
HTR6 P50406 1/20 0.33
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32
PSENEN Q9NZ42 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2570026 0.92 F10 (0.35) CCKBRF10ROCK2CA12CA1
SCHEMBL2569424 0.91 CCKBR (0.39) CCKBRF10ROCK2ALDH1A1POLB
SCHEMBL2567238 0.91 CCKBR (0.38) CCKBRF10ROCK2ALDH1A1POLB
SCHEMBL3382049 0.91 CCKBR (0.35) CCKBRF10ROCK2ALDH1A1NPSR1
SCHEMBL2571203 0.90 F10 (0.34) CCKBRF10ROCK2ALDH1A1PSEN1
SCHEMBL2574207 0.90 CCKBR (0.38) CCKBRF10ROCK2CA12CA1
SCHEMBL2573538 0.90 CCKBR (0.38) CCKBRF10ROCK2
SCHEMBL2572736 0.89 CCKBR (0.38) CCKBRF10ROCK2ALDH1A1POLB
SCHEMBL3382957 0.89 F10 (0.44) CCKBRF10ROCK2DRD2HTR2C
SCHEMBL2571105 0.89 KDM4E (0.34) CCKBRF10ROCK2ALDH1A1PSEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899330-B1 SUBSTITUTED GLYCINAMIDES HAVING AN ANTITHROMBOTIC AND FACTOR XA-INHIBITING EFFECT BOEHRINGER INGELHEIM INT (DE) 2010-11-24 EP disclosed