SCHEMBL3380869

SCHEMBL3380869

O=C(C[C@H]1CCCc2c1cnn2-c1ccccc1)N1CCOCC1

nearest known ligand 0.66

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.66
TMEM97 Q5BJF2 1/20 0.66
LMNA P02545 1/20 0.46
DHODH Q02127 4/20 0.45
ALDH1A1 P00352 3/20 0.44
HSP90AA1 P07900 1/20 0.43
MAPK1 P28482 1/20 0.43
ADAM10 O14672 1/20 0.42
ERBB2 P04626 1/20 0.42
MMP2 P08253 1/20 0.42
FKBP1A P62942 1/20 0.42
POLB P06746 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3354308 1.00 SIGMAR1 (0.66) SIGMAR1TMEM97LMNADHODHALDH1A1
SCHEMBL3354305 1.00 SIGMAR1 (0.66) SIGMAR1TMEM97LMNADHODHALDH1A1
SCHEMBL959673 0.90 TMEM97 (0.55) SIGMAR1TMEM97DHODHADAM10ERBB2
SCHEMBL3378446 0.83 SIGMAR1 (0.58) SIGMAR1TMEM97DHODHKMT2A
SCHEMBL3379565 0.83 SIGMAR1 (0.58) SIGMAR1TMEM97DHODHKMT2A
SCHEMBL955851 0.83 SIGMAR1 (0.58) SIGMAR1TMEM97DHODHKMT2A
Oxalic Acid SCHEMBL955643 0.82 SIGMAR1 (0.90) SIGMAR1TMEM97DHODHALDH1A1HSP90AA1
SCHEMBL3383254 0.80 SIGMAR1 (1.00) SIGMAR1TMEM97DHODHALDH1A1HSP90AA1
SCHEMBL3381500 0.80 SIGMAR1 (1.00) SIGMAR1TMEM97DHODHALDH1A1HSP90AA1
SCHEMBL954332 0.80 SIGMAR1 (1.00) SIGMAR1TMEM97DHODHALDH1A1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010066829-A1 PROCESS FOR OBTAINING ENANTIOMERICALLY ENRICHED PYRAZOLE DERIVATIVES LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2010-06-17 WO disclosed
WO-2010066829-A1 PROCESS FOR OBTAINING ENANTIOMERICALLY ENRICHED PYRAZOLE DERIVATIVES LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2010-06-17 WO disclosed
EP-2196458-A1 Process for obtaining enantiomerically enriched pyrazole derivatives Laboratorios Del. Dr. Esteve, S.A. (ES) 2010-06-16 EP disclosed
EP-2196458-A1 Process for obtaining enantiomerically enriched pyrazole derivatives Laboratorios Del. Dr. Esteve, S.A. (ES) 2010-06-16 EP disclosed