SCHEMBL3383407

SCHEMBL3383407

CC(C)(C)c1cc(NC(=O)CCc2ccc(-c3cnc4cc(-c5ccc(S(C)(=O)=O)cc5)ccn34)cc2)[nH]n1

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 12/20 0.47
KDR P35968 6/20 0.45
FGFR3 P22607 2/20 0.42
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3383393 0.87 FLT3 (0.47) FLT3KDRFGFR3
SCHEMBL3195720 0.85 FLT3 (0.50) FLT3KDRFGFR3KCNH2
SCHEMBL3383188 0.85 FLT3 (0.48) FLT3KDRFGFR3
SCHEMBL3381104 0.82 KDR (0.55) FLT3KDRFGFR3KCNH2
SCHEMBL3385924 0.81 FLT3 (0.44) FLT3KDRFGFR3
SCHEMBL27705869 0.81 KDR (0.49) FLT3KDRFGFR3
SCHEMBL3197333 0.80 FLT3 (0.53) FLT3KDRKCNH2
SCHEMBL3195685 0.79 KDR (0.54) FLT3KDRFGFR3
SCHEMBL3385811 0.77 KDR (0.49) FLT3KDRFGFR3
SCHEMBL3385731 0.75 KDR (0.50) FLT3KDRFGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed